SCHEMBL29928245

SCHEMBL29928245

COc1cc2ccnc(-n3nc(N)nc3N)c2cc1OC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 9/20 0.49
PIK3CA P42336 1/20 0.47
PIK3CB P42338 1/20 0.47
MTOR P42345 1/20 0.47
PRKDC P78527 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.46
MAPT P10636 2/20 0.46
GAA P10253 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.43
CYP3A4 P08684 3/20 0.42
PDE10A Q9Y233 3/20 0.42
USP2 O75604 2/20 0.42
ALDH1A1 P00352 2/20 0.42
LMNA P02545 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C9 P11712 2/20 0.42
MAPK1 P28482 2/20 0.42
CYP2C19 P33261 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29927676 0.78 ATM (0.69) ATMPIK3CAPIK3CBMTORPRKDC
SCHEMBL29927588 0.74 AXL (0.51) ATMPIK3CAPIK3CBMTORPRKDC
SCHEMBL15595899 0.73 SMN1; SMN2 (0.57) SMN1; SMN2MAPTGAATDP1L3MBTL1
SCHEMBL29929117 0.72 SMN1; SMN2 (0.55) ATMPIK3CAPIK3CBMTORPRKDC
SCHEMBL4236664 0.72 AXL (0.77)
SCHEMBL4774035 0.69 ACHE (0.60) SMN1; SMN2CYP3A4USP2ALDH1A1LMNA
SCHEMBL29928526 0.69 HTR2C (0.46) ALDH1A1KDM4E
SCHEMBL2919337 0.69 NCF1 (0.60) MAPTCYP3A4USP2ALDH1A1CYP1A2
SCHEMBL3974591 0.68 CYP3A4 (0.54) SMN1; SMN2MAPTGAATDP1L3MBTL1
SCHEMBL30458203 0.68 CYP3A4 (0.54) SMN1; SMN2MAPTGAATDP1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110551105-B Substituted triazoles useful as AXL inhibitors 里格尔制药公司 2022-10-18 CN claimed
CN-110551105-B Substituted triazoles useful as AXL inhibitors 里格尔制药公司 2022-10-18 CN disclosed