SCHEMBL29930508

SCHEMBL29930508

C[Si](C)(C)CCOCn1nc(-c2cncnc2)c2cc(Br)cnc21

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 3/20 0.36
DYRK1A Q13627 1/20 0.34
DYRK1B Q9Y463 1/20 0.34
MERTK Q12866 2/20 0.33
PDE10A Q9Y233 1/20 0.31
MAPT P10636 1/20 0.30
PDE1B Q01064 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1592834 0.88 MERTK (0.39) DGAT1DYRK1ADYRK1BMERTK
SCHEMBL29930809 0.87 DGAT1 (0.37) DGAT1DYRK1ADYRK1BMERTKMAPT
SCHEMBL29930401 0.87 DYRK1B (0.40) DGAT1DYRK1BMERTKPDE1B
SCHEMBL29930779 0.86 AXL (0.41) DGAT1DYRK1ADYRK1BMERTKMAPT
SCHEMBL29930917 0.84 DYRK1B (0.38) DGAT1DYRK1BMERTK
SCHEMBL29935301 0.83 DGAT1 (0.33) DGAT1DYRK1B
SCHEMBL29930407 0.83 DYRK1B (0.39) DGAT1DYRK1BMERTKPDE1B
SCHEMBL29113927 0.82 DGAT1 (0.36) DGAT1
SCHEMBL29930775 0.82 MAPT (0.35) DGAT1MAPT
SCHEMBL29930815 0.82 AXL (0.41) DGAT1DYRK1BMERTKMAPTPDE1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022235097-A1 PHARMACEUTICAL COMPOSITION CONTAINING NOVEL PYRAZOLO[3,4-B]PYRIDINE DERIVATIVE FOR PREVENTION OR TREATMENT OF METABOLIC DISEASE INCLUDING OBESITY AND DIABETES MELLITUS OR NONALCOHOLIC STEATOHEPATITIS 한국화학연구원 2022-11-10 WO disclosed