SCHEMBL29930648

SCHEMBL29930648

O=C(O)N1CCC2(CC1)Cc1cccnc1C2

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SPR P35270 1/20 0.42
ALDH1A1 P00352 11/20 0.40
CYP3A4 P08684 9/20 0.40
CYP2C9 P11712 7/20 0.40
MAPK1 P28482 5/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CHRM2 P08172 1/20 0.40
HSD17B10 Q99714 11/20 0.40
CYP2C19 P33261 7/20 0.40
HPGD P15428 6/20 0.40
CYP1A2 P05177 6/20 0.40
CYP2D6 P10635 6/20 0.40
USP2 O75604 2/20 0.40
TSHR P16473 6/20 0.39
HIF1A Q16665 1/20 0.39
HRH3 Q9Y5N1 1/20 0.38
ALOX15 P16050 1/20 0.37
HSD11B1 P28845 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29550671 0.81 HRH3 (0.50) ALDH1A1CYP3A4CYP2C9MAPK1SMN1; SMN2
SCHEMBL8316507 0.81 HRH3 (0.50) ALDH1A1CYP3A4CYP2C9MAPK1SMN1; SMN2
SCHEMBL13004992 0.81 POLB (0.50) ALDH1A1CYP3A4MAPK1HSD17B10CYP2C19
SCHEMBL22958207 0.80 TSHR (0.36) CYP2C9CHRM2CYP2C19CYP1A2CYP2D6
SCHEMBL30179224 0.80 SPR (0.33) SPRALDH1A1CYP3A4CYP2C9MAPK1
SCHEMBL30486552 0.79 SIGMAR1 (0.38) SPRALDH1A1SMN1; SMN2CHRM2HSD17B10
SCHEMBL27454475 0.79 AVPR1A (0.35) SPRALDH1A1CYP3A4CYP2C9MAPK1
SCHEMBL30486670 0.79 AVPR1A (0.35) SPRALDH1A1CYP3A4CYP2C9MAPK1
SCHEMBL30179411 0.78 SPR (0.32) SPRALDH1A1CYP3A4CYP2C9MAPK1
SCHEMBL29637622 0.76 ABHD6 (0.36) ALDH1A1CYP3A4CYP2C9MAPK1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113493440-B Salt of nitrogen-containing heteroaromatic derivative and crystal form thereof 上海翰森生物医药科技有限公司 2024-08-23 CN disclosed
CN-115052866-B Crystal form of nitrogen-containing heteroaromatic derivative free alkali 上海翰森生物医药科技有限公司 2024-06-25 CN disclosed
CN-115353509-B Nitrogen-containing heteroaromatic derivative regulator, preparation method and application thereof 江苏豪森药业集团有限公司 2024-04-12 CN disclosed
EP-4227307-A1 PYRAZOLOPYRAZINE COMPOUNDS AS SHP2 INHIBITORS Genzyme Corporation (US) 2023-08-16 EP disclosed
US-20230242551-A1 ISOTOPE-SUBSTITUTED SPIRO AROMATIC RING COMPOUND AND APPLICATION THEREOF ETERN BIOPHARMA (SHANGHAI) CO., LTD. (CN) 2023-08-03 US disclosed
EP-4166549-A1 ISOTOPE-SUBSTITUTED SPIRO AROMATIC RING COMPOUND AND APPLICATION THEREOF Etern Biopharma (Shanghai) Co., Ltd. (CN) 2023-04-19 EP disclosed
CN-115353509-A Aza-containing aromatic derivative regulator, preparation method and application thereof 江苏豪森药业集团有限公司 2022-11-18 CN disclosed
CN-111295374-B Aza-containing aromatic derivative regulator, preparation method and application thereof 江苏豪森药业集团有限公司 2022-11-04 CN disclosed
CN-115052866-A Crystal form of free base of nitrogen-containing heteroaromatic derivative 上海翰森生物医药科技有限公司 2022-09-13 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230242551-A1 ISOTOPE-SUBSTITUTED SPIRO AROMATIC RING COMPOUND AND APPLICATION THEREOF SLCO1B1, SLCO1B3, SLCO2B1 SPR 189/4885ALDH1A1 884/4885CYP3A4 35/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.