SCHEMBL2993065

SCHEMBL2993065

O=c1cc[nH]c2cc([N+](=O)[O-])ccc12

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.56
DAO P14920 1/20 0.56
PARP1 P09874 3/20 0.53
GRIA1 P42261 1/20 0.50
GRIA2 P42262 1/20 0.50
GRIA3 P42263 1/20 0.50
GRIA4 P48058 1/20 0.50
HSD17B10 Q99714 1/20 0.50
PKM P14618 1/20 0.49
PKLR P30613 1/20 0.49
CYP3A4 P08684 1/20 0.47
NAMPT P43490 1/20 0.47
XDH P47989 1/20 0.47
CA12 O43570 2/20 0.45
CA9 Q16790 2/20 0.45
PTPRA P18433 1/20 0.44
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
RAB9A P51151 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2980781 0.86 CA12 (0.53) ALDH1A1DAOPARP1GRIA1GRIA2
SCHEMBL8600209 0.81 DAO (0.50) ALDH1A1DAOPARP1GRIA1GRIA2
SCHEMBL30011 0.77 MAPT (0.54) ALDH1A1DAOPARP1GRIA1GRIA2
SCHEMBL29904251 0.77 MAPT (0.54) ALDH1A1DAOPARP1GRIA1GRIA2
SCHEMBL29236590 0.76 PKM (0.56) DAOPARP1GRIA1GRIA2GRIA3
SCHEMBL915292 0.76 ALDH1A1 (0.50) ALDH1A1DAOPARP1GRIA1GRIA2
SCHEMBL8487610 0.74 TDP1 (0.50) ALDH1A1DAOGRIA1GRIA2GRIA3
SCHEMBL6008297 0.74 PARP1 (0.73) ALDH1A1DAOPARP1GRIA1GRIA2
SCHEMBL29993384 0.74 PARP1 (0.73) ALDH1A1DAOPARP1GRIA1GRIA2
SCHEMBL1664417 0.73 CYP3A4 (0.66) ALDH1A1DAOPARP1GRIA1GRIA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100173332-A1 Method for the Fluorescent Detection of Nitroreductase Activity Using Nitro-Substituted Aromatic Compounds AUCKLAND UNISERVICES LIMITED 2010-07-08 US disclosed
WO-2008030120-A1 A METHOD FOR THE FLUORESCENT DETECTION OF NITROREDUCTASE ACTIVITY USING NITRO-SUBSTITUTED AROMATIC COMPOUNDS AUCKLAND UNISERVICES LIMITED (NZ) 2008-03-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100173332-A1 Method for the Fluorescent Detection of Nitroreductase Activity Using Nitro-Substituted Aromatic Compounds BLVRB, POR, CBR3 ALDH1A1 119/4885DAO 310/4885PARP1 3775/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.