SCHEMBL29934262

SCHEMBL29934262

CC1=C(C)C(=O)N(Nc2cc(Cl)c3cccc(Br)c3n2)C1=O

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
XPO1 O14980 3/20 0.56
ALDH1A1 P00352 1/20 0.40
MAPT P10636 3/20 0.34
GAA P10253 1/20 0.34
ENPP3 O14638 1/20 0.34
ENPP1 P22413 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
P2RX7 Q99572 1/20 0.33
CRHR1 P34998 1/20 0.33
PARP1 P09874 1/20 0.33
LMNA P02545 1/20 0.32
EGFR P00533 1/20 0.32
PDE7A Q13946 1/20 0.31
GRM2 Q14416 1/20 0.31
ADORA1 P30542 1/20 0.31
HRH4 Q9H3N8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1592549 1.00 XPO1 (0.56) XPO1ALDH1A1MAPTGAAENPP3
SCHEMBL1592361 0.88 XPO1 (0.67) XPO1MAPTL3MBTL1SMN1; SMN2CRHR1
SCHEMBL1592533 0.87 XPO1 (0.59) XPO1MAPTGAAL3MBTL1SMN1; SMN2
SCHEMBL1592551 0.84 XPO1 (0.38) XPO1ALDH1A1MAPTGAAENPP3
SCHEMBL1592387 0.81 XPO1 (0.53) XPO1ALDH1A1MAPTL3MBTL1
SCHEMBL1592940 0.77 XPO1 (0.46) XPO1MAPT
SCHEMBL1592575 0.73 LMNA (0.51) XPO1ALDH1A1MAPTSMN1; SMN2LMNA
SCHEMBL1592535 0.72 XPO1 (0.41) XPO1MAPTGAAL3MBTL1SMN1; SMN2
SCHEMBL1592523 0.72 XPO1 (1.00) XPO1PARP1
SCHEMBL23872048 0.72 XPO1 (0.52) XPO1ALDH1A1MAPTGAAP2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4074704-A1 QUINOLINE COMPOUNDS WITH ANTI-CANCER ACTIVITY CanBas Co., Ltd. (JP) 2022-10-19 EP disclosed