Dequalinium

Dequalinium

SCHEMBL2993904

Cc1cc(N)c2ccccc2[n+]1CCCCCCCCCC[n+]1c(C)cc(N)c2ccccc21.[Br-].[Br-]

nearest known ligand 0.97

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHKACHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGHRH2OPRM1

The experimentally established mechanism targets of Dequalinium. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 known ✓ P08172 1/20 0.97
CHRM1 known ✓ P11229 1/20 0.97
ACHE known ✓ P22303 1/20 0.97
OPRM1 known ✓ P35372 1/20 0.97
PRKCA P17252 13/20 0.97
MEN1 O00255 4/20 0.97
GMNN O75496 4/20 0.97
LMNA P02545 4/20 0.97
POLB P06746 4/20 0.97
MAPT P10636 4/20 0.97
APEX1 P27695 4/20 0.97
RECQL P46063 4/20 0.97
BLM P54132 4/20 0.97
PMP22 Q01453 4/20 0.97
KMT2A Q03164 4/20 0.97
SMN1; SMN2 Q16637 4/20 0.97
NPSR1 Q6W5P4 4/20 0.97
TDP1 Q9NUW8 4/20 0.97
ALDH1A1 P00352 3/20 0.97
TP53 P04637 3/20 0.97

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6305111 0.98 PRKCA (1.00) PRKCAMEN1GMNNLMNAPOLB
Dequalinium SCHEMBL29557297 0.98 PRKCA (1.00) PRKCAMEN1GMNNLMNAPOLB
Dequalinium SCHEMBL29577841 0.98 PRKCA (1.00) PRKCAMEN1GMNNLMNAPOLB
Dequalinium SCHEMBL149457 0.98 PRKCA (1.00) PRKCAMEN1GMNNLMNAPOLB
SCHEMBL6299633 0.98 PRKCA (1.00) PRKCAMEN1GMNNLMNAPOLB
SCHEMBL6298118 0.98 PRKCA (1.00) PRKCAMEN1GMNNLMNAPOLB
Dequalinium SCHEMBL1008339 0.97 PRKCA (0.97) PRKCAMEN1GMNNLMNAPOLB
Dequalinium SCHEMBL2335922 0.97 PRKCA (1.00) PRKCAMEN1GMNNLMNAPOLB
Dequalinium SCHEMBL2544854 0.97 MEN1 (1.00) PRKCAMEN1GMNNLMNAPOLB
Dequalinium SCHEMBL34043 0.97 MEN1 (1.00) PRKCAMEN1GMNNLMNAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230414570-A1 COMPOSITIONS AGAINST CANDIDA INFECTIONS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2023-12-28 US disclosed
US-11793790-B2 Compositions against Candida infections UNIVERSITEIT ANTWERPEN (BE) 2023-10-24 US disclosed
EP-3949962-B1 COMPOSITIONS AGAINST CANDIDA INFECTIONS UNIV LEUVEN KATH (BE) 2023-09-13 EP disclosed
EP-3949962-A1 COMPOSITIONS AGAINST CANDIDA INFECTIONS Katholieke Universiteit Leuven (BE) 2022-02-09 EP disclosed
EP-3654973-B1 COMPOSITIONS AGAINST CANDIDA INFECTIONS UNIV LEUVEN KATH (BE) 2021-08-18 EP disclosed
EP-3654973-A1 COMPOSITIONS AGAINST CANDIDA INFECTIONS Katholieke Universiteit Leuven (BE) 2020-05-27 EP disclosed
US-20200138786-A1 COMPOSITIONS AGAINST CANDIDA INFECTIONS UNIVERSITEIT ANTWERPEN (BE) 2020-05-07 US disclosed
WO-2019015975-A1 COMPOSITIONS AGAINST CANDIDA INFECTIONS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2019-01-24 WO disclosed
US-8071640-B2 Urea oligomers, their preparation process and pharmaceutical compositions containing them CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2011-12-06 US disclosed
US-20100184849-A1 UREA OLIGOMERS, THEIR PREPARATION PROCESS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQU (FR) 2010-07-22 US disclosed
US-7691899-B2 Urea oligomers, the preparation method thereof and pharmaceutical composition containing same CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2010-04-06 US disclosed
US-20050038105-A1 Novel urea oligomers, the preparation method thereof and pharmaceutical composition containing same CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2005-02-17 US disclosed
WO-1996023050-A1 CLEANSING COMPOSITIONS JEYES GROUP PLC (GB) 1996-08-01 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100184849-A1 UREA OLIGOMERS, THEIR PREPARATION PROCESS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM UACA, RAN, URB2 CHRM2 2902/4885CHRM1 2581/4885ACHE 1131/4885
US-20050038105-A1 Novel urea oligomers, the preparation method thereof and pharmaceutical composition containing same URB2, NOXO1, UACA CHRM2 3836/4885CHRM1 3276/4885ACHE 2850/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.