SCHEMBL29944809

SCHEMBL29944809

O=C(OCc1ccccc1)N1CC(Nc2nc(Cl)nc3[nH]cc(Cl)c23)C2(CC2)C1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 5/20 0.37
ATXN2 Q99700 2/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
JAK2 O60674 2/20 0.36
JAK1 P23458 2/20 0.36
USP30 Q70CQ3 1/20 0.35
GRIN2B Q13224 3/20 0.35
CYP2C19 P33261 1/20 0.35
OPRK1 P41145 2/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
OPRD1 P41143 1/20 0.34
KDM1A O60341 1/20 0.34
MAPT P10636 1/20 0.34
TYK2 P29597 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29944772 0.92 ENPP2 (0.39) ENPP2ATXN2MEN1KMT2ANPSR1
SCHEMBL29944949 0.82 JAK3 (0.55) JAK3
SCHEMBL30305650 0.77 JAK3 (0.49) ENPP2JAK3
SCHEMBL22609913 0.77 JAK3 (0.49) ENPP2JAK3
SCHEMBL29944802 0.76 JAK3 (0.56) JAK3
SCHEMBL30948974 0.75 GRM5 (0.44) ENPP2ATXN2MEN1KMT2ANPSR1
SCHEMBL31634701 0.75 GRM5 (0.44) ENPP2ATXN2MEN1KMT2ANPSR1
SCHEMBL30210344 0.74 SMN1; SMN2 (0.48) ENPP2ATXN2MEN1KMT2ANPSR1
SCHEMBL31634718 0.73 RAB9A (0.44) ENPP2ATXN2MEN1KMT2ANPSR1
SCHEMBL30948981 0.73 RAB9A (0.44) ENPP2ATXN2MEN1KMT2ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115244055-B Pyrimidine five-membered ring derivative and application thereof 江苏先声药业有限公司 2024-09-03 CN disclosed
CN-115244055-A Pyrimido five-membered ring derivative and application thereof 江苏先声药业有限公司 2022-10-25 CN disclosed