SCHEMBL29948217

SCHEMBL29948217

CCc1nc(N)ncc1Br

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 1/20 0.41
DHFR P00374 5/20 0.40
GRM4 Q14833 1/20 0.39
HSP90AA1 P07900 1/20 0.38
HEXA P06865 4/20 0.37
HEXB P07686 4/20 0.37
MEN1 O00255 1/20 0.35
SLC22A1 O15245 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
HTR1A P08908 1/20 0.35
ADRA2A P08913 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
HTR2A P28223 1/20 0.35
ADRA1A P35348 1/20 0.35
HTR2B P41595 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23534954 1.00 NUDT1 (0.41) NUDT1DHFRGRM4HSP90AA1HEXA
SCHEMBL27559232 0.79 GRM4 (0.39) NUDT1GRM4HSP90AA1
SCHEMBL22834670 0.79 LMNA (0.40) NUDT1GRM4HSP90AA1MEN1LMNA
SCHEMBL29652037 0.79 LMNA (0.40) NUDT1GRM4HSP90AA1MEN1LMNA
SCHEMBL10399566 0.78 NUDT1 (0.43) NUDT1DHFRHSP90AA1HEXAHEXB
SCHEMBL27559431 0.78 NUDT1 (0.40) NUDT1GRM4HSP90AA1
SCHEMBL18031204 0.77 NUDT1 (0.59) NUDT1GRM4HSP90AA1HEXAHEXB
SCHEMBL28150953 0.77 DHFR (0.49) NUDT1DHFRHSP90AA1
SCHEMBL232075 0.75 NUDT1 (0.41) NUDT1DHFRHSP90AA1HEXAHEXB
SCHEMBL233104 0.75 NUDT1 (0.42) NUDT1DHFRGRM4HSP90AA1HEXA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4077282-A1 PRMT5 INHIBITORS Merck Sharp & Dohme LLC (US) 2022-10-26 EP disclosed
EP-4076459-A1 PRMT5 INHIBITORS Merck Sharp & Dohme LLC (US) 2022-10-26 EP disclosed