SCHEMBL29948277

SCHEMBL29948277

CN(C)C(=O)C1CN1S(=O)(=O)c1ccc2c(C=O)c(N(C)C)ccc2c1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.41
MME P08473 2/20 0.36
ACE P12821 2/20 0.36
ECE1 P42892 2/20 0.36
ERN1 O75460 2/20 0.35
PKM P14618 1/20 0.35
CCR4 P51679 10/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.34
ALDH1A1 P00352 2/20 0.34
LMNA P02545 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
F2 P00734 1/20 0.34
F10 P00742 1/20 0.34
KDM4E B2RXH2 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23630319 1.00 CASP3 (0.41) CASP3MMEACEECE1ERN1
SCHEMBL23630332 0.88 ALDH1A1 (0.42) CASP3MMEACEECE1ALDH1A1
SCHEMBL29948321 0.84 CASP3 (0.43) CASP3MMEACEECE1PKM
SCHEMBL23630364 0.84 CASP3 (0.43) CASP3MMEACEECE1PKM
SCHEMBL23630309 0.72 KDM4E (0.39) ERN1ALDH1A1LMNAKDM4EHTT
SCHEMBL29948225 0.72 KDM4E (0.39) ERN1ALDH1A1LMNAKDM4EHTT
SCHEMBL23630483 0.71 KMT2A (0.50) CASP3ALDH1A1LMNASMN1; SMN2HTT
SCHEMBL23630363 0.71 ALDH1A1 (0.44) CASP3MMEACEECE1CCR4
SCHEMBL30225533 0.69 KMT2A (0.46) F2HTT
SCHEMBL23630601 0.68 CCR4 (0.40) CASP3CCR4LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4087651-A1 AROMATIC SULPHONAMIDES DERIVATIVES THAT INHIBITS PDI A1, THEIR SYNTHESIS AND USE UNIWERSYTET JAGIELLONSKI (PL) 2022-11-16 EP claimed
EP-4087651-A1 AROMATIC SULPHONAMIDES DERIVATIVES THAT INHIBITS PDI A1, THEIR SYNTHESIS AND USE UNIWERSYTET JAGIELLONSKI (PL) 2022-11-16 EP disclosed