SCHEMBL29952702

SCHEMBL29952702

[C-]#[N+]Cc1c(C)cc(C)cc1C

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.36
RAPGEF4 Q8WZA2 2/20 0.35
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
HTR1D P28221 1/20 0.33
HTR1B P28222 1/20 0.33
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
GAA P10253 1/20 0.30
MAPT P10636 1/20 0.30
MEN1 O00255 1/20 0.30
MAPK1 P28482 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12629117 0.72 PGK1 (0.38)
SCHEMBL29954468 0.72 IDH1 (0.35) CYP11B1CYP11B2ALDH1A1
SCHEMBL1316919 0.69 HTR1D (0.48) HRH3RAPGEF4CYP11B1CYP11B2HTR1D
SCHEMBL27995904 0.69 HRH3 (0.54) HRH3RAPGEF4CYP11B1CYP11B2HTR1D
SCHEMBL12032123 0.69 HRH3 (0.32) HRH3RAPGEF4CYP11B1CYP11B2HTR1D
SCHEMBL327084 0.67 HRH3 (0.41) HRH3RAPGEF4CYP11B1CYP11B2HTR1D
SCHEMBL28489168 0.67 HRH3 (0.41) HRH3RAPGEF4CYP11B1CYP11B2HTR1D
SCHEMBL29951023 0.67 PGK1 (0.38) ALDH1A1
SCHEMBL29953337 0.65 TAAR1 (0.50) KDM4EALDH1A1LMNAGAAMAPT
Bromide SCHEMBL17647120 0.65 RAPGEF4 (0.46) HRH3RAPGEF4CYP11B1CYP11B2HTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed