SCHEMBL29954439

SCHEMBL29954439

COc1cc(C=O)c2cc[nH]c2n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38
MAPT P10636 1/20 0.38
ADORA1 P30542 2/20 0.37
PDCD1 Q15116 2/20 0.36
CD274 Q9NZQ7 2/20 0.36
ATR Q13535 2/20 0.36
ATRIP Q8WXE1 2/20 0.36
CHEK1 O14757 1/20 0.36
MCL1 Q07820 1/20 0.36
DYRK1A Q13627 2/20 0.35
CLK1 P49759 1/20 0.35
CLK2 P49760 1/20 0.35
CLK3 P49761 1/20 0.35
CDK5 Q00535 1/20 0.35
CDK5R1 Q15078 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
DYRK1B Q9Y463 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29722091 0.79 TRPA1 (0.38) CYP1A2ADORA1PDCD1CD274ATR
SCHEMBL23147607 0.79 TRPA1 (0.38) CYP1A2ADORA1PDCD1CD274ATR
SCHEMBL16612853 0.77 BRD4 (0.43) ALDH1A1KDM4EADORA1PDCD1CD274
SCHEMBL29957561 0.76 DYRK1A (0.38) CYP1A2ADORA1DYRK1AADORA2AKMT2A
SCHEMBL26106331 0.76 DYRK1A (0.38) ALDH1A1KDM4EMAPTADORA1PDCD1
SCHEMBL30611953 0.76 DYRK1A (0.38) ALDH1A1KDM4EMAPTADORA1PDCD1
SCHEMBL3360828 0.76 PRKCI (0.44) ADORA1PDCD1CD274ATRATRIP
SCHEMBL23148049 0.76 AXL (0.44) ADORA1PDCD1CD274ATRATRIP
SCHEMBL23152002 0.71 LMNA (0.48) ALDH1A1KDM4ECYP1A2MAPTMCL1
SCHEMBL29935837 0.71 LMNA (0.48) ALDH1A1KDM4ECYP1A2MAPTMCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed