SCHEMBL2995628

SCHEMBL2995628

CC(C)C(C)(c1ccc(OCc2nccs2)cc1)c1ccc(-c2nnn(C)n2)cc1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
NFKB1 P19838 1/20 0.46
NFKB2 Q00653 1/20 0.46
RELA Q04206 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
NPSR1 Q6W5P4 2/20 0.37
ACACB O00763 1/20 0.37
MAOB P27338 2/20 0.35
ALOX5AP P20292 1/20 0.35
TSHR P16473 1/20 0.33
MAPK1 P28482 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3000148 0.89 AOC3 (0.41) NPC1RAB9ASMN1; SMN2NPSR1MAOB
SCHEMBL2990099 0.88 NPC1 (0.45) NPC1RAB9ANFKB1NFKB2RELA
SCHEMBL2993029 0.83 NPC1 (0.52) NPC1RAB9ANFKB1NFKB2RELA
SCHEMBL2245990 0.81 ALOX5AP (0.54) NPC1RAB9ANFKB1NFKB2RELA
SCHEMBL3002980 0.78 APP (0.45) RAB9AACACBALOX5APL3MBTL1
SCHEMBL3000902 0.77 ALOX5AP (0.43) NPC1RAB9ASMN1; SMN2ACACBALOX5AP
SCHEMBL2993269 0.77 NR4A2 (0.49) NPC1RAB9ASMN1; SMN2ACACBMAPK1
SCHEMBL3000188 0.76 ACACB (0.46) RAB9AACACBMAOBALOX5AP
Ammonia Solution, Strong SCHEMBL2997486 0.76 ACACB (0.37) ACACBALOX5AP
SCHEMBL2995463 0.76 AOC3 (0.39) ACACBALOX5AP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2546232-A1 Diphenyl Substituted Alkanes Merck Sharp & Dohme Corp. (US) 2013-01-16 EP disclosed
US-20100190761-A1 DIPHENYL SUBSTITUTED ALKANES MERCK SHARP & DOHME CORP. 2010-07-29 US disclosed
EP-2170065-A1 DIPHENYL SUBSTITUTED ALKANES Merck Sharp & Dohme Corp. (US) 2010-04-07 EP disclosed
WO-2008156721-A1 DIPHENYL SUBSTITUTED ALKANES MERCK & CO., INC. (US) 2008-12-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100190761-A1 DIPHENYL SUBSTITUTED ALKANES ALOX5, ALOX15, ALOX15B NPC1 603/4885RAB9A 4316/4885NFKB1 145/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.