SCHEMBL29965256

SCHEMBL29965256

O=c1[nH]c2cc(CO)ccc2n2c(Br)ccc12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 9/20 0.42
PDE9A O76083 5/20 0.41
PDE5A O76074 4/20 0.40
TP53 P04637 1/20 0.38
CDC7 O00311 1/20 0.38
PLK4 O00444 1/20 0.38
AURKA O14965 1/20 0.38
MAPK13 O15264 1/20 0.38
PDPK1 O15530 1/20 0.38
DYRK3 O43781 1/20 0.38
PRKD3 O94806 1/20 0.38
MAP4K4 O95819 1/20 0.38
PAK4 O96013 1/20 0.38
ERBB2 P04626 1/20 0.38
NTRK1 P04629 1/20 0.38
PRKCG P05129 1/20 0.38
FYN P06241 1/20 0.38
CSF1R P07333 1/20 0.38
RET P07949 1/20 0.38
IGF1R P08069 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28895087 0.77 PARP1 (0.46) PARP1PDE9APDE5ATP53AURKA
SCHEMBL3337877 0.74 PARP1 (0.51) PARP1PDE9APDE5ATP53MAP4K4
SCHEMBL29965987 0.74 PDE5A (0.45) PARP1PDE9APDE5ATP53PLA2G10
SCHEMBL29966010 0.73 PARP1 (0.66) PARP1TP53CDC7PLK4AURKA
SCHEMBL30273139 0.72 PARP1 (0.41) PARP1PDE9ACDC7PLK4AURKA
SCHEMBL28895268 0.72 ALDH1A1 (0.55) PARP1PLK4DYRK3PRKD3MAP4K4
SCHEMBL29965925 0.72 ALDH1A1 (0.55) PARP1PLK4DYRK3PRKD3MAP4K4
SCHEMBL16174315 0.69 LMNA (0.51) PARP1TP53DAO
SCHEMBL31195706 0.69 PARP1 (0.33) PARP1PDE9APDE5ACDC7PLK4
SCHEMBL29965714 0.68 PARP1 (0.51) PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115368362-A Quinoxalinone derivatives as BTK inhibitors and application thereof 华东理工大学 2022-11-22 CN disclosed