SCHEMBL29968376

SCHEMBL29968376

O=C(O)Cc1ccc(Cn2c(-c3ccccc3)nc3c(-c4ccc(C5=CCCCC5)cc4)cccc32)cc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PPARG P37231 5/20 0.41
P2RX3 P56373 3/20 0.40
PDE6D O43924 1/20 0.39
ALDH1A1 P00352 1/20 0.39
ALDH2 P05091 1/20 0.39
ALDH3A1 P30838 1/20 0.39
TP53 P04637 1/20 0.39
FBP1 P09467 1/20 0.39
HRH3 Q9Y5N1 1/20 0.37
ABCC4 O15439 1/20 0.37
LMNA P02545 1/20 0.37
GAA P10253 1/20 0.37
TSHR P16473 1/20 0.37
PTGS1 P23219 1/20 0.37
HTT P42858 1/20 0.37
CNR2 P34972 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29967886 0.98 PPARG (0.40) PPARGP2RX3PDE6DALDH1A1ALDH2
SCHEMBL29967492 0.94 TP53 (0.39) PPARGP2RX3PDE6DALDH1A1ALDH2
SCHEMBL29968184 0.91 PPARG (0.43) PPARGP2RX3PDE6DALDH1A1ALDH2
SCHEMBL29967971 0.90 PPARG (0.42) PPARGP2RX3
SCHEMBL29967905 0.90 P2RX3 (0.38) PPARGP2RX3TP53FBP1GAA
SCHEMBL29967514 0.90 CNR2 (0.37) PPARGP2RX3TP53HRH3GAA
SCHEMBL29968167 0.89 NR1H4 (0.44) PPARGP2RX3HRH3
SCHEMBL29967824 0.87 KDM4E (0.49) CNR2
SCHEMBL29967830 0.86 PLA2G10 (0.42) PPARGP2RX3TP53
SCHEMBL29967497 0.84 PPARG (0.42) PPARGALDH1A1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260165-B Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2024-08-06 CN disclosed
CN-115260165-A Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2022-11-01 CN disclosed