SCHEMBL29967971

SCHEMBL29967971

Cc1nc2c(-c3ccc(C4=CCCCC4)cc3)cccc2n1Cc1ccc(CC(=O)O)cc1

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PPARG P37231 6/20 0.42
P2RX3 P56373 5/20 0.41
DCTPP1 Q9H773 1/20 0.38
AGTR1 P30556 2/20 0.38
AGTR2 P50052 2/20 0.38
PTAFR P25105 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29967912 0.93 P2RX3 (0.39) PPARGP2RX3DCTPP1
SCHEMBL29967886 0.92 PPARG (0.40) PPARGP2RX3
SCHEMBL29968376 0.90 PPARG (0.41) PPARGP2RX3
SCHEMBL29968012 0.90 NR1H4 (0.46) PPARGP2RX3DCTPP1AGTR1AGTR2
SCHEMBL29968433 0.89 CYP19A1 (0.39) PPARGP2RX3AGTR1AGTR2
SCHEMBL29968198 0.88 DCTPP1 (0.42) PPARGP2RX3DCTPP1AGTR1AGTR2
SCHEMBL29967688 0.88 CNR2 (0.38) PPARGP2RX3
SCHEMBL29968232 0.86 PDE10A (0.40) PPARGP2RX3DCTPP1AGTR1AGTR2
SCHEMBL29967953 0.86 PLA2G10 (0.41) PPARGP2RX3DCTPP1
SCHEMBL29967938 0.85 PPARG (0.42) PPARGP2RX3AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260165-B Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2024-08-06 CN disclosed
CN-115260165-A Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2022-11-01 CN disclosed