SCHEMBL29967905

SCHEMBL29967905

O=C(O)Cc1cccc(Cn2c(-c3cccc(CC(=O)O)c3)nc3c(-c4ccc(C5=CCCCC5)cc4)cccc32)c1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 4/20 0.38
TP53 P04637 2/20 0.37
MAPT P10636 1/20 0.37
PPARG P37231 3/20 0.36
CNR2 P34972 2/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
PTGER4 P35408 1/20 0.35
PTGIR P43119 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.34
KDM4E B2RXH2 1/20 0.34
GAA P10253 1/20 0.34
CCR2 P41597 1/20 0.34
FBP1 P09467 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29967492 0.96 TP53 (0.39) P2RX3TP53MAPTPPARGCNR2
SCHEMBL29967912 0.91 P2RX3 (0.39) P2RX3PPARGCNR2PTGDR2
SCHEMBL29968376 0.90 PPARG (0.41) P2RX3TP53PPARGCNR2GAA
SCHEMBL29967886 0.90 PPARG (0.40) P2RX3TP53PPARGFBP1
SCHEMBL29967574 0.88 PPARG (0.41) P2RX3TP53MAPTPPARGCCR2
SCHEMBL29967830 0.86 PLA2G10 (0.42) P2RX3TP53MAPTPPARGCCR2
SCHEMBL29967971 0.84 PPARG (0.42) P2RX3PPARG
SCHEMBL29967514 0.84 CNR2 (0.37) P2RX3TP53PPARGCNR2PTGDR2
SCHEMBL29968184 0.83 PPARG (0.43) P2RX3PPARG
SCHEMBL29968167 0.82 NR1H4 (0.44) P2RX3PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115260165-B Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2024-08-06 CN disclosed
CN-115260165-A Benzo nitrogen-containing five-membered heterocyclic compound and synthesis and application thereof 中国科学院上海药物研究所 2022-11-01 CN disclosed