SCHEMBL2997143

SCHEMBL2997143

N#Cc1[nH]c2ccc(Br)cc2c1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSNK2A1 P68400 2/20 0.44
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
MAPT P10636 2/20 0.39
CHUK O15111 1/20 0.39
GPR84 Q9NQS5 1/20 0.39
AR P10275 1/20 0.38
NPSR1 Q6W5P4 2/20 0.38
PRNP P04156 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
PPARG P37231 1/20 0.38
HIF1A Q16665 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
NR2E3 Q9Y5X4 1/20 0.38
NCOR2 Q9Y618 1/20 0.38
JAK2 O60674 2/20 0.37
CHEK1 O14757 1/20 0.37
AURKA O14965 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15486057 0.79 CSNK2A1 (0.44) CSNK2A1LMNAHPGDMAPTCHUK
SCHEMBL2729876 0.79 KDM4E (0.42) MAPTCHUKGPR84CLK2DYRK1A
SCHEMBL22206950 0.78 PIM1 (0.44) LMNAHPGDMAPTRXFP1JAK2
SCHEMBL16920116 0.76 CSNK2A1 (0.41) CSNK2A1LMNAHPGDMAPTCHUK
SCHEMBL2730451 0.76 KDM4E (0.56) HPGDMAPTCHUKGPR84RXFP1
SCHEMBL11622624 0.74 ALDH1A1 (0.54) CSNK2A1LMNAMAPTNPSR1RXFP1
SCHEMBL2731190 0.74 DRD2 (0.47) LMNAHPGDCYP1A2DYRK1AMEN1
SCHEMBL4489319 0.72 PRNP (0.51) CSNK2A1HPGDMAPTNPSR1PRNP
SCHEMBL14689247 0.71 CHUK (0.57) CSNK2A1LMNAHPGDMAPTCHUK
SCHEMBL29366993 0.70 CHUK (0.64) LMNAHPGDMAPTCHUKGPR84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100197687-A1 Indoles Useful in the Treatment of Inflammation BIOLIPOX AB (SE) 2010-08-05 US disclosed
EP-1841736-A1 INDOLES USEFUL IN THE TREATMENT OF INFLAMMATION Biolipox AB (SE) 2007-10-10 EP disclosed
WO-2006077367-A1 INDOLES USEFUL IN THE TREATMENT OF INFLAMATION BIOLIPOX AB (SE) 2006-07-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100197687-A1 Indoles Useful in the Treatment of Inflammation IDO1, IDO2, TPH1 CSNK2A1 834/4885LMNA 3796/4885HPGD 337/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.