SCHEMBL29977295

SCHEMBL29977295

Nc1nc2ccccc2c2c1ncn2Cc1cccc(CN2CCCC2=O)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 7/20 0.48
PDE4D Q08499 2/20 0.48
LMNA P02545 1/20 0.48
POLB P06746 1/20 0.48
HRH2 P25021 1/20 0.48
ADRA1D P25100 1/20 0.48
HTR2A P28223 1/20 0.48
ADORA2A P29274 1/20 0.48
ADRA1A P35348 1/20 0.48
NUDT1 P36639 1/20 0.48
HTR2B P41595 1/20 0.48
KCNH2 Q12809 1/20 0.48
NLRP3 Q96P20 5/20 0.45
L3MBTL1 Q9Y468 1/20 0.43
TLR8 Q9NR97 3/20 0.40
MAOB P27338 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
PDE4A P27815 1/20 0.39
PDE4B Q07343 1/20 0.39
PDE4C Q08493 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29809072 0.89 L3MBTL1 (0.46) KCNH2L3MBTL1MAOBSMN1; SMN2PDE4A
SCHEMBL24732579 0.84 TLR7 (0.54) TLR7PDE4DLMNAPOLBHRH2
SCHEMBL29808887 0.84 TLR7 (0.54) TLR7PDE4DLMNAPOLBHRH2
SCHEMBL3188618 0.80 TLR7 (0.67) TLR7PDE4DLMNAPOLBHRH2
SCHEMBL29976933 0.79 TLR7 (0.54) TLR7PDE4DLMNAPOLBHRH2
SCHEMBL29809062 0.79 NLRP3 (0.52) TLR7KCNH2NLRP3L3MBTL1TLR8
SCHEMBL24732755 0.79 NLRP3 (0.52) TLR7KCNH2NLRP3L3MBTL1TLR8
SCHEMBL24732578 0.79 HRH3 (0.50) TLR7PDE4DLMNAPOLBHRH2
Hydrochloric Acid SCHEMBL3197884 0.79 TLR7 (0.66) TLR7PDE4DLMNAPOLBHRH2
SCHEMBL24732765 0.76 TLR7 (0.57) TLR7PDE4DLMNAPOLBHRH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022161420-A1 CLASS OF HETEROAROMATIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 上海翊石医药科技有限公司 2022-08-04 WO disclosed