SCHEMBL29977949

SCHEMBL29977949

O=C(Nc1cccnc1)N1CCc2cc(-c3noc(C(F)(F)F)n3)sc2C1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 2/20 0.51
HDAC6 Q9UBN7 2/20 0.51
HTR2C P28335 14/20 0.45
HTR2A P28223 12/20 0.45
PDGFRB P09619 1/20 0.44
TRPV1 Q8NER1 1/20 0.42
CYP1A2 P05177 2/20 0.42
HTR2B P41595 3/20 0.42
MEN1 O00255 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
MAPT P10636 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
KMT2A Q03164 1/20 0.42
HDAC1 Q13547 1/20 0.41
HDAC8 Q9BY41 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29978684 0.93 HDAC4 (0.51) HDAC4HDAC6HTR2CHTR2APDGFRB
SCHEMBL29977979 0.91 HDAC4 (0.47) HDAC4HDAC6CYP1A2MEN1CYP3A4
SCHEMBL29977806 0.90 HDAC6 (0.37) HDAC4HDAC6HDAC1HDAC8
SCHEMBL29978286 0.87 CYP3A4 (0.44) HDAC4HDAC6TRPV1CYP1A2MEN1
SCHEMBL29978167 0.87 HDAC6 (0.46) HDAC4HDAC6MAPTHDAC1HDAC8
SCHEMBL29979015 0.86 MEN1 (0.47) HDAC4HDAC6TRPV1MEN1MAPT
SCHEMBL29977966 0.86 NAMPT (0.43) HDAC4HDAC6TRPV1MAPT
SCHEMBL29978402 0.86 NPC1 (0.47) HDAC4HDAC6CYP1A2MEN1CYP3A4
SCHEMBL29978706 0.86 HPGD (0.49) HDAC4HDAC6PDGFRBHDAC1HDAC8
SCHEMBL29978688 0.85 RAB9A (0.46) HDAC4HDAC6MAPTHDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022234470-A1 NOVEL FUSED HETEROCYCLIC COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI PI INDUSTRIES LTD. (IN) 2022-11-10 WO claimed
WO-2022234470-A1 NOVEL FUSED HETEROCYCLIC COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI PI INDUSTRIES LTD. (IN) 2022-11-10 WO disclosed