SCHEMBL29977966

SCHEMBL29977966

O=C(Nc1ccc(C(F)(F)F)cc1)N1CCc2cc(-c3noc(C(F)(F)F)n3)sc2C1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 2/20 0.43
EPHX2 P34913 1/20 0.42
KCNH2 Q12809 1/20 0.42
CACNA1C Q13936 1/20 0.42
TRPV1 Q8NER1 6/20 0.41
HDAC4 P56524 3/20 0.41
HDAC6 Q9UBN7 1/20 0.41
TRPM8 Q7Z2W7 4/20 0.40
HPGDS O60760 1/20 0.40
KDM4E B2RXH2 1/20 0.39
MAPT P10636 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29978402 0.93 NPC1 (0.47) NAMPTHDAC4HDAC6TRPM8MAPT
SCHEMBL29979015 0.93 MEN1 (0.47) NAMPTTRPV1HDAC4HDAC6KDM4E
SCHEMBL29978389 0.93 NAMPT (0.46) NAMPTEPHX2KCNH2CACNA1CTRPV1
SCHEMBL29978688 0.92 RAB9A (0.46) NAMPTHDAC4HDAC6MAPT
SCHEMBL29977979 0.92 HDAC4 (0.47) HDAC4HDAC6
SCHEMBL29977836 0.91 KMT2A (0.39) HDAC4HDAC6MAPT
SCHEMBL29978134 0.90 EPHX2 (0.45) NAMPTEPHX2TRPV1TRPM8KDM4E
SCHEMBL29979201 0.89 GPR142 (0.45) TRPV1HDAC4HDAC6MAPTNPSR1
SCHEMBL29977806 0.88 HDAC6 (0.37) HDAC4HDAC6
SCHEMBL29978286 0.87 CYP3A4 (0.44) TRPV1HDAC4HDAC6MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022234470-A1 NOVEL FUSED HETEROCYCLIC COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI PI INDUSTRIES LTD. (IN) 2022-11-10 WO claimed
WO-2022234470-A1 NOVEL FUSED HETEROCYCLIC COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI PI INDUSTRIES LTD. (IN) 2022-11-10 WO disclosed