SCHEMBL29978286

SCHEMBL29978286

O=C(Nc1cccc(F)c1)N1CCc2cc(-c3noc(C(F)(F)F)n3)sc2C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 7/20 0.44
USP2 O75604 6/20 0.44
CYP2C9 P11712 2/20 0.44
HIF1A Q16665 1/20 0.44
CYP1A2 P05177 2/20 0.43
LMNA P02545 2/20 0.43
MAPT P10636 2/20 0.43
HTT P42858 2/20 0.43
NPSR1 Q6W5P4 1/20 0.43
HDAC4 P56524 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
MEN1 O00255 1/20 0.42
RECQL P46063 1/20 0.42
KMT2A Q03164 1/20 0.42
CYP2C19 P33261 2/20 0.42
HDAC8 Q9BY41 2/20 0.42
HDAC6 Q9UBN7 2/20 0.42
HDAC1 Q13547 1/20 0.42
TRPV1 Q8NER1 1/20 0.41
NPC1 O15118 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29978228 0.93 CYP3A4 (0.44) CYP3A4USP2CYP2C9HIF1ACYP1A2
SCHEMBL29978070 0.92 HDAC4 (0.41) CYP3A4USP2CYP2C9HIF1ACYP1A2
SCHEMBL29977979 0.91 HDAC4 (0.47) CYP3A4USP2CYP2C9CYP1A2LMNA
SCHEMBL29978402 0.91 NPC1 (0.47) CYP3A4CYP2C9CYP1A2LMNAMAPT
SCHEMBL29978488 0.89 NPC1 (0.39) LMNAMAPTHTTHDAC4SMN1; SMN2
SCHEMBL29977949 0.87 HDAC4 (0.51) CYP3A4CYP2C9CYP1A2MAPTHDAC4
SCHEMBL29979015 0.87 MEN1 (0.47) LMNAMAPTHTTNPSR1HDAC4
SCHEMBL29977966 0.87 NAMPT (0.43) MAPTNPSR1HDAC4HDAC6TRPV1
SCHEMBL29979201 0.86 GPR142 (0.45) CYP3A4LMNAMAPTHTTNPSR1
SCHEMBL29978688 0.86 RAB9A (0.46) MAPTHDAC4SMN1; SMN2HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022234470-A1 NOVEL FUSED HETEROCYCLIC COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI PI INDUSTRIES LTD. (IN) 2022-11-10 WO claimed
WO-2022234470-A1 NOVEL FUSED HETEROCYCLIC COMPOUNDS FOR COMBATING PHYTOPATHOGENIC FUNGI PI INDUSTRIES LTD. (IN) 2022-11-10 WO disclosed