SCHEMBL2999475

SCHEMBL2999475

C/C(C(N)=O)=C(/C)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LDHA P00338 2/20 0.50
LDHB P07195 1/20 0.50
LMNA P02545 3/20 0.44
BLM P54132 2/20 0.44
ALOX15 P16050 1/20 0.44
PMP22 Q01453 1/20 0.44
TDP1 Q9NUW8 2/20 0.42
ACHE P22303 1/20 0.38
FFAR3 O14843 1/20 0.38
LCK P06239 1/20 0.38
FYN P06241 1/20 0.38
CRBN Q96SW2 1/20 0.32
ALDH1A1 P00352 1/20 0.31
OR51E2 Q9H255 1/20 0.31
THRB P10828 1/20 0.31
FNTA P49354 1/20 0.31
FNTB P49356 1/20 0.31
PGGT1B P53609 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL343159 1.00 LDHA (0.50) LDHALDHBLMNABLMALOX15
SCHEMBL343160 1.00 LDHA (0.50) LDHALDHBLMNABLMALOX15
SCHEMBL27696587 0.86 LMNA (0.58) LDHALDHBLMNABLMALOX15
SCHEMBL4141273 0.86 LMNA (0.58) LDHALDHBLMNABLMALOX15
SCHEMBL4779556 0.86 LMNA (0.58) LDHALDHBLMNABLMALOX15
SCHEMBL27476647 0.82 LMNA (0.54) LDHALDHBLMNABLMALOX15
SCHEMBL105998 0.82 FFAR3 (0.55) LDHALDHBLMNABLMALOX15
SCHEMBL10661655 0.82 FFAR3 (0.55) LDHALDHBLMNABLMALOX15
SCHEMBL141678 0.82 FFAR3 (0.55) LDHALDHBLMNABLMALOX15
SCHEMBL10661623 0.82 FFAR3 (0.55) LDHALDHBLMNABLMALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20190119415-A1 GRAFT COPOLYMER FOR CATION-EXCHANGE CHROMATOGRAPHY MERCK PATENT GMBH (DE) 2019-04-25 US claimed
EP-2152405-B2 GRAFT COPOLYMER FOR CATION-EXCHANGE CHROMATOGRAPHY MERCK PATENT GMBH (DE) 2017-04-05 EP claimed
EP-2152405-B1 GRAFT COPOLYMER FOR CATION-EXCHANGE CHROMATOGRAPHY MERCK PATENT GMBH (DE) 2012-10-17 EP claimed
US-20190119415-A1 GRAFT COPOLYMER FOR CATION-EXCHANGE CHROMATOGRAPHY MERCK PATENT GMBH (DE) 2019-04-25 US disclosed
EP-2152405-B2 GRAFT COPOLYMER FOR CATION-EXCHANGE CHROMATOGRAPHY MERCK PATENT GMBH (DE) 2017-04-05 EP disclosed
US-20140183136-A1 GRAFT COPOLYMER FOR CATION-EXCHANGE CHROMATOGRAPHY MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2014-07-03 US disclosed
EP-2152405-B1 GRAFT COPOLYMER FOR CATION-EXCHANGE CHROMATOGRAPHY MERCK PATENT GMBH (DE) 2012-10-17 EP disclosed
US-20100181254-A1 GRAFT COPOLYMER FOR CATION- EXCHANGE CHROMATOGRAPHY MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2010-07-22 US disclosed
EP-2152405-A1 GRAFT COPOLYMER FOR CATION-EXCHANGE CHROMATOGRAPHY Merck Patent GmbH (DE) 2010-02-17 EP disclosed
WO-2008145270-A1 GRAFT COPOLYMER FOR CATION-EXCHANGE CHROMATOGRAPHY MERCK PATENT GMBH (DE) 2008-12-04 WO disclosed
EP-0503301-B1 Peptide derivatives and application thereof FUJI PHOTO FILM CO LTD (JP) 1997-11-26 EP disclosed
EP-0619118-B1 Use of peptide derivatives FUJI PHOTO FILM CO LTD (JP) 1997-06-11 EP disclosed
US-5436221-A Oligopeptides as antitumor agents FUJI PHOTO FILM CO., LTD. (JP) 1995-07-25 US disclosed
EP-0619118-A1 Use of peptide derivatives FUJI PHOTO FILM CO., LTD. (JP) 1994-10-12 EP disclosed
EP-0503301-A2 Peptide derivatives and application thereof FUJI PHOTO FILM CO., LTD. (JP) 1992-09-16 EP disclosed