SCHEMBL30002556

SCHEMBL30002556

COc1cc(F)c(N)cc1OCc1c(F)ccc2ccncc12

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAOA P21397 2/20 0.39
MAPT P10636 7/20 0.38
GAA P10253 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
KIT P10721 1/20 0.37
KDR P35968 2/20 0.35
FLT1 P17948 1/20 0.35
PDE10A Q9Y233 1/20 0.35
PDPK1 O15530 1/20 0.35
RET P07949 1/20 0.34
KIF5B P33176 1/20 0.34
CLK1 P49759 1/20 0.34
DYRK1A Q13627 1/20 0.34
PLAU P00749 1/20 0.34
ERBB2 P04626 1/20 0.34
EPHA2 P29317 1/20 0.34
TRPA1 O75762 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28892234 1.00 MAOA (0.39) MAOAMAPTGAASMN1; SMN2TDP1
SCHEMBL30002412 0.88 MAOA (0.40) MAOAMAPTGAASMN1; SMN2TDP1
SCHEMBL28892522 0.88 MAOA (0.40) MAOAMAPTGAASMN1; SMN2TDP1
SCHEMBL30002702 0.85 KIT (0.37) MAOAMAPTGAASMN1; SMN2TDP1
SCHEMBL28892670 0.85 KIT (0.37) MAOAMAPTGAASMN1; SMN2TDP1
SCHEMBL28892526 0.83 SCN1A (0.47) MAOAMAPTGAASMN1; SMN2TDP1
SCHEMBL30002548 0.83 SCN1A (0.47) MAOAMAPTGAASMN1; SMN2TDP1
SCHEMBL28892434 0.82 KDR (0.37) MAOAMAPTGAASMN1; SMN2TDP1
SCHEMBL30002084 0.82 KDR (0.37) MAOAMAPTGAASMN1; SMN2TDP1
SCHEMBL28959518 0.82 LMNA (0.42) MAOAMAPTGAATDP1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115232144-B Nitrogen-containing condensed ring derivative, pharmaceutical composition, and preparation method and application thereof 长春金赛药业有限责任公司 2024-04-02 CN disclosed
CN-115232144-A Nitrogen-containing fused ring derivative, pharmaceutical composition, preparation method and application thereof 长春金赛药业有限责任公司 2022-10-25 CN disclosed