SCHEMBL30003169

SCHEMBL30003169

[2H]c1nc(N)cc2cc(Br)ccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 2/20 0.48
KDM4E B2RXH2 1/20 0.45
MEN1 O00255 1/20 0.45
ALDH1A1 P00352 1/20 0.45
MAPT P10636 1/20 0.45
KMT2A Q03164 1/20 0.45
CYP2A6 P11509 1/20 0.39
GSK3A P49840 1/20 0.36
CDK9 P50750 1/20 0.36
CDK5 Q00535 1/20 0.36
TAOK1 Q7L7X3 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
HTT P42858 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36
PDPK1 O15530 1/20 0.35
PABPC1 P11940 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35
TYMS P04818 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19516842 1.00 BACE1 (0.48) BACE1KDM4EMEN1ALDH1A1MAPT
SCHEMBL558436 0.80 PDPK1 (0.57) BACE1KDM4EMEN1ALDH1A1MAPT
SCHEMBL30381711 0.80 PDPK1 (0.57) BACE1KDM4EMEN1ALDH1A1MAPT
SCHEMBL558012 0.76 PDPK1 (0.57) BACE1KDM4EMEN1ALDH1A1MAPT
SCHEMBL30676520 0.76 PDPK1 (0.57) BACE1KDM4EMEN1ALDH1A1MAPT
SCHEMBL30381549 0.76 PDPK1 (0.57) BACE1KDM4EMEN1ALDH1A1MAPT
Methylene Chloride SCHEMBL27807255 0.74 PDPK1 (0.50) BACE1KDM4EMEN1ALDH1A1MAPT
SCHEMBL29371678 0.68 CYP2A6 (0.72) BACE1KDM4EMEN1ALDH1A1MAPT
SCHEMBL2051640 0.68 CYP2A6 (0.72) BACE1KDM4EMEN1ALDH1A1MAPT
SCHEMBL30579926 0.68 CYP2A6 (0.41) BACE1KDM4EMEN1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260022108-A1 ISOQUINOLIN-3-YL CARBOXAMIDES AND PREPARATION AND USE THEREOF TENARX, INC. 2026-01-22 US disclosed
EP-4559905-A2 ISOQUINOLIN-3-YL CARBOXAMIDES AS WNT INHIBITORS BioSplice Therapeutics, Inc. (US) 2025-05-28 EP disclosed
US-12281097-B2 Isoquinolin-3-yl carboxamides and preparation and use thereof BIOSPLICE THERAPEUTICS, INC. (US) 2025-04-22 US disclosed
US-11673881-B2 Isoquinolin-3-yl carboxamides and preparation and use thereof BIOSPLICE THERAPEUTICS, INC. (US) 2023-06-13 US disclosed
US-20230104155-A1 ISOQUINOLIN-3-YL CARBOXAMIDES AND PREPARATION AND USE THEREOF VICKERS-SPLICE CO-INVESTMENT LLC (KY) 2023-04-06 US disclosed
US-11548872-B2 Isoquinolin-3-yl carboxamides and preparation and use thereof BIOSPLICE THERAPEUTICS, INC. (US) 2023-01-10 US disclosed
CN-109311819-B Isoquinolin-3-yl carboxamides, their preparation and their use 萨穆梅德有限公司 2022-10-25 CN disclosed
US-20220332698-A1 ISOQUINOLIN-3-YL CARBOXAMIDES AND PREPARATION AND USE THEREOF TENARX, INC. 2022-10-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12281097-B2 Isoquinolin-3-yl carboxamides and preparation and use thereof WNT1, WNT3, WNT3A BACE1 1926/4885KDM4E 1534/4885MEN1 4429/4885
US-11673881-B2 Isoquinolin-3-yl carboxamides and preparation and use thereof DYRK1A, DYRK3, DYRK1B BACE1 1111/4885KDM4E 1528/4885MEN1 4483/4885
US-11548872-B2 Isoquinolin-3-yl carboxamides and preparation and use thereof WNT1, WNT3, WNT3A BACE1 1926/4885KDM4E 1534/4885MEN1 4429/4885
US-20230104155-A1 ISOQUINOLIN-3-YL CARBOXAMIDES AND PREPARATION AND USE THEREOF DYRK1A, DYRK3, DYRK1B BACE1 1111/4885KDM4E 1528/4885MEN1 4483/4885
US-20260022108-A1 ISOQUINOLIN-3-YL CARBOXAMIDES AND PREPARATION AND USE THEREOF WNT1, WNT3, WNT3A BACE1 2628/4885KDM4E 2457/4885MEN1 4709/4885
US-20220332698-A1 ISOQUINOLIN-3-YL CARBOXAMIDES AND PREPARATION AND USE THEREOF WNT1, WNT3, WNT3A BACE1 1926/4885KDM4E 1534/4885MEN1 4429/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.