SCHEMBL30005644

SCHEMBL30005644

COC(=O)c1cc(CN(CCN(C)C(=O)OC(C)(C)C)C(=O)OC(C)(C)C)ccc1N(C)S(C)(=O)=O

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.36
ALDH1A1 P00352 3/20 0.34
HTT P42858 1/20 0.34
HDAC1 Q13547 3/20 0.34
HDAC3 O15379 2/20 0.34
HDAC2 Q92769 2/20 0.34
NCOR2 Q9Y618 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
POLB P06746 1/20 0.32
MCOLN3 Q8TDD5 1/20 0.32
CYP19A1 P11511 2/20 0.32
KDM4E B2RXH2 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
ALOX15 P16050 1/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30005928 0.90 HDAC1 (0.35) KMT2AALDH1A1HDAC1HDAC3HDAC2
SCHEMBL30006749 0.84 KMT2A (0.45) KMT2AL3MBTL1ALDH1A1CYP19A1KDM4E
SCHEMBL30006097 0.79 PARP1 (0.38) KMT2AALDH1A1HDAC1HDAC3HDAC2
SCHEMBL30006618 0.77 CA1 (0.38) KMT2AALDH1A1HDAC1HDAC3HDAC2
SCHEMBL30005739 0.77 KMT2A (0.50) KMT2AL3MBTL1ALDH1A1HDAC1GAA
SCHEMBL30964962 0.72 GLS (0.40) KMT2AL3MBTL1ALDH1A1HTTSMN1; SMN2
SCHEMBL14012666 0.72 HSP90AA1 (0.42) HDAC1HDAC3HDAC2NCOR2
SCHEMBL3118579 0.71 GLS (0.39) KMT2AALDH1A1HTTHDAC1HDAC3
SCHEMBL3110201 0.71 GLS (0.43) KMT2AALDH1A1HTTHDAC1HDAC3
SCHEMBL1323637 0.71 ALDH1A1 (0.58) ALDH1A1HTTSMN1; SMN2KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022220725-A1 LPXH INHIBITORS AS ANTI-INFECTIVE AGENTS ZAMARATSKI EDOUARD (SE) 2022-10-20 WO disclosed