SCHEMBL30007554

SCHEMBL30007554

CC(C)S(=O)(=O)c1ccc(-c2cnc3[nH]cc(C(=O)N4CCC(c5ccccc5)CC4)c3c2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 1/20 0.47
AXL P30530 1/20 0.46
CAMKK2 Q96RR4 4/20 0.42
SGK1 O00141 3/20 0.42
PIK3CA P42336 1/20 0.42
AURKA O14965 1/20 0.42
CAMKK1 Q8N5S9 1/20 0.42
SGK3 Q96BR1 1/20 0.42
SGK2 Q9HBY8 1/20 0.42
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
IL2 P60568 1/20 0.41
MAP4K1 Q92918 1/20 0.41
PAK1 Q13153 3/20 0.40
AAK1 Q2M2I8 1/20 0.40
IKBKB O14920 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30007265 0.91 AVPR1A (0.49) AVPR1AAXLCAMKK2SGK1PIK3CA
SCHEMBL30007738 0.85 KDM5A (0.42) CA12CA1CA2CA7CA9
SCHEMBL30007804 0.82 ALDH1A1 (0.46) AXLMAP3K11
SCHEMBL30007369 0.82 DRD2 (0.47) CAMKK2SGK1IL2MAP4K1IKBKB
SCHEMBL30007672 0.82 PAK1 (0.53) AXLCAMKK2PIK3CACA1CA2
SCHEMBL30007824 0.82 CHRM2 (0.44) PIK3CAMAP4K1PAK1MAP3K11CHRM2
Hydrochloric Acid SCHEMBL30007576 0.79 AXL (0.54) AXLCAMKK2SGK1PIK3CAAURKA
SCHEMBL30008314 0.76 AXL (0.67) AXLCAMKK2SGK1PIK3CAAAK1
SCHEMBL30007677 0.75 AXL (0.50) AXLCAMKK2SGK1PIK3CAAAK1
SCHEMBL30007560 0.75 CA12 (0.43) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022237922-A1 ANTITUMOR COMPOUNDS BASED ON NITROGEN HETEROCYCLES AND USE THEREOF AS MEDICAMENTS FAKULTNI NEMOCNICE HRADEC KRALOVE (CZ) 2022-11-17 WO disclosed