SCHEMBL30007265

SCHEMBL30007265

CS(=O)(=O)c1ccc(-c2cnc3[nH]cc(C(=O)N4CCC(c5ccccc5)CC4)c3c2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AVPR1A P37288 1/20 0.49
AXL P30530 1/20 0.48
PAK1 Q13153 3/20 0.45
CAMKK2 Q96RR4 4/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
SGK1 O00141 2/20 0.44
PIK3CA P42336 1/20 0.44
AURKA O14965 1/20 0.44
CAMKK1 Q8N5S9 1/20 0.44
SGK3 Q96BR1 1/20 0.44
SGK2 Q9HBY8 1/20 0.44
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43
IL2 P60568 1/20 0.43
MAP4K1 Q92918 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30007554 0.91 AVPR1A (0.47) AVPR1AAXLPAK1CAMKK2SGK1
SCHEMBL30007560 0.84 CA12 (0.43) CA12CA1CA2CA7CA9
SCHEMBL30007741 0.81 CA12 (0.44) CA12CA1CA2CA7CA9
Hydrochloric Acid SCHEMBL30007736 0.78 CAMKK2 (0.57) AXLPAK1CAMKK2CYP2C9CYP2C19
SCHEMBL30007738 0.75 KDM5A (0.42) CA12CA1CA2CA7CA9
SCHEMBL30007360 0.74 AXL (0.72) AXLPAK1CAMKK2CYP2C9CYP2C19
SCHEMBL30007824 0.72 CHRM2 (0.44) PAK1CYP2C9CYP2C19PIK3CAMAP4K1
SCHEMBL30007804 0.72 ALDH1A1 (0.46) AXLCYP2C9CYP2C19MAP3K11
SCHEMBL30007672 0.72 PAK1 (0.53) AXLPAK1CAMKK2CYP2C9CYP2C19
SCHEMBL30007369 0.72 DRD2 (0.47) CAMKK2SGK1IL2MAP4K1MAP3K11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022237922-A1 ANTITUMOR COMPOUNDS BASED ON NITROGEN HETEROCYCLES AND USE THEREOF AS MEDICAMENTS FAKULTNI NEMOCNICE HRADEC KRALOVE (CZ) 2022-11-17 WO claimed
WO-2022237922-A1 ANTITUMOR COMPOUNDS BASED ON NITROGEN HETEROCYCLES AND USE THEREOF AS MEDICAMENTS FAKULTNI NEMOCNICE HRADEC KRALOVE (CZ) 2022-11-17 WO disclosed