SCHEMBL30014728

SCHEMBL30014728

COc1ccc(COc2ccccc2S(=O)(=O)NC2(CS(C)(=O)=O)CC2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 1/20 0.42
ADRA1D P25100 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
NCOR2 Q9Y618 1/20 0.41
ABCB1 P08183 2/20 0.41
CYP19A1 P11511 1/20 0.41
PTGDR2 Q9Y5Y4 1/20 0.39
TP53 P04637 1/20 0.39
ALDH1A1 P00352 2/20 0.38
LMNA P02545 1/20 0.38
MAPK1 P28482 1/20 0.38
BCHE P06276 2/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29965183 0.79 CYP19A1 (0.35) CYP19A1TP53ALDH1A1LMNAMAPK1
SCHEMBL29965415 0.73 NPC1 (0.54) HTR1AADRA1DADRA1AADRA1BNPC1
SCHEMBL6567074 0.71 ALDH1A1 (0.52) ABCB1ALDH1A1BCHEMEN1KMT2A
SCHEMBL16018989 0.69 ABCB1 (0.68) HTR1AADRA1DADRA1AADRA1BNPC1
Water SCHEMBL8980729 0.66 RXRA (0.52) NPC1RAB9AABCB1TP53HTT
SCHEMBL12358221 0.66 NPC1 (0.65) HTR1AADRA1DADRA1AADRA1BNPC1
SCHEMBL12465690 0.65 ALDH1A1 (0.48) HTR1AADRA1DADRA1AADRA1BNPC1
SCHEMBL30449333 0.65 CYP19A1 (0.56) HTR1AADRA1DADRA1AADRA1BNPC1
SCHEMBL22193705 0.65 ABCB1 (0.70) HTR1AADRA1DADRA1AADRA1BNPC1
SCHEMBL12301149 0.64 ABCB1 (0.60) HTR1AADRA1DADRA1AADRA1BNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115244037-A Substituted triazinones as thyroid hormone receptor agonists 上海诚益生物科技有限公司 2022-10-25 CN disclosed