SCHEMBL30023637

SCHEMBL30023637

Cc1ccc(CC2CO2)c(Cc2ccccc2)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC5A2 P31639 4/20 0.44
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C19 P33261 2/20 0.43
TSHR P16473 1/20 0.43
BCL2 P10415 1/20 0.40
BCL2L1 Q07817 1/20 0.40
CHRM2 P08172 1/20 0.37
CHRM5 P08912 1/20 0.37
CHRM3 P20309 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GLA P06280 1/20 0.37
MGLL Q99685 2/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
ALOX5 P09917 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4442750 0.80 BCL2 (0.54) CYP3A4CYP2D6CYP2C19TSHRBCL2
SCHEMBL9066731 0.77 BCL2 (0.50) CYP3A4CYP2D6CYP2C19TSHRBCL2
SCHEMBL3301748 0.75 CYP3A4 (0.53) CYP3A4CYP2D6CYP2C19TSHRBCL2
SCHEMBL1276089 0.75 CYP3A4 (0.57) CYP3A4CYP2D6CYP2C19TSHRBCL2
SCHEMBL607838 0.74 BCL2 (0.47) CYP3A4CYP2D6CYP2C19TSHRBCL2
SCHEMBL5879437 0.74 LMNA (0.40) TSHRALDH1A1GLAL3MBTL1
SCHEMBL31438264 0.73 ALDH1A1 (0.48) CYP2D6TSHRCHRM2ALDH1A1GLA
SCHEMBL7049331 0.73 ALDH1A1 (0.48) CYP2D6TSHRCHRM2ALDH1A1GLA
SCHEMBL28335494 0.73 ALDH1A1 (0.48) CYP2D6TSHRCHRM2ALDH1A1GLA
SCHEMBL4958841 0.72 TP53 (0.37) ALDH1A1MEN1KMT2ASMN1; SMN2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115243764-B Heterocyclic derivatives as TRMP antagonists 奇华顿股份有限公司 2025-01-03 CN disclosed
EP-4114523-A1 HETEROCYCLIC DERIVATIVES AS TRMP8 ANTAGONISTS Givaudan SA (CH) 2023-01-11 EP disclosed
CN-115243764-A Heterocyclic derivatives as TRMP8 antagonists 奇华顿股份有限公司 2022-10-25 CN disclosed