SCHEMBL300261

SCHEMBL300261

[CH]c1c(CCC)noc1C

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26867970 0.74 CYP1A2 (0.33) CYP1A2CYP2C9
SCHEMBL11527632 0.67 GPX4 (0.42)
SCHEMBL2428653 0.65 MLYCD (0.33) CYP1A2CYP2C9
SCHEMBL14923174 0.65 CYP1A2 (0.33) CYP1A2CYP2C9
SCHEMBL285589 0.65 ALDH1A1 (0.44)
SCHEMBL8995000 0.64 TLR8 (0.38)
SCHEMBL20843963 0.64
SCHEMBL8237746 0.64 LMNA (0.44) CYP1A2CYP2C9
SCHEMBL15255830 0.63 TLR8 (0.34)
SCHEMBL14923170 0.63 CYP1A2 (0.32) CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427457-A1 ISOXAZOLE-PYRIDINE DERIVATIVES AS GABA MODULATORS F. Hoffmann-La Roche AG (CH) 2012-03-14 EP disclosed
WO-2010127978-A1 ISOXAZOLE-PYRIDINE DERIVATIVES AS GABA MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2010-11-11 WO disclosed