SCHEMBL300407

SCHEMBL300407

COc1cnc2[nH]cc(-c3c(C=O)cccc3[N+](=O)[O-])c2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 3/20 0.40
NEK1 Q96PY6 1/20 0.40
KIT P10721 4/20 0.39
CYP19A1 P11511 1/20 0.38
AXL P30530 3/20 0.38
DYRK1A Q13627 3/20 0.38
DYRK3 O43781 2/20 0.38
ROCK2 O75116 2/20 0.38
PRKD3 O94806 2/20 0.38
MAP4K4 O95819 2/20 0.38
CDK1 P06493 2/20 0.38
MARK3 P27448 2/20 0.38
FLT4 P35916 2/20 0.38
FLT3 P36888 2/20 0.38
SYK P43405 2/20 0.38
CSNK1D P48730 2/20 0.38
CLK2 P49760 2/20 0.38
GSK3A P49840 2/20 0.38
GSK3B P49841 2/20 0.38
BLK P51451 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL300124 0.86 AXL (0.39) KITAXLDYRK1AGSK3BCDK5
SCHEMBL300130 0.83 MTNR1A (0.43) NTRK1NEK1KITAXLDYRK1A
SCHEMBL1713918 0.73 ALDH1A1 (0.55) NTRK1NEK1KITDYRK1ACSF1R
SCHEMBL27530428 0.70 ERN1 (0.49) CYP19A1
SCHEMBL8141976 0.69 MTNR1A (0.44) DYRK1ASYKEGFRMTNR1AMTNR1B
SCHEMBL31451378 0.69 MTNR1A (0.44) DYRK1ASYKEGFRMTNR1AMTNR1B
SCHEMBL1716453 0.69 POLB (0.53) CYP19A1MTNR1AMTNR1B
SCHEMBL300129 0.67 MAOB (0.49)
SCHEMBL10638535 0.67 MEN1 (0.45) CYP19A1
SCHEMBL298453 0.66 AAK1 (0.49) NEK1AXLIRAK4MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427433-A1 SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS Plexxikon, Inc. (US) 2012-03-14 EP disclosed
WO-2010129570-A1 SOLID FORMS OF SULFONAMIDES AND AMINO ACIDS PLEXXIKON, INC. (US) 2010-11-11 WO disclosed