SCHEMBL30050418

SCHEMBL30050418

COc1ccc2cnccc2c1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 8/20 0.60
CYP11B1 P15538 7/20 0.60
CYP17A1 P05093 3/20 0.59
CYP19A1 P11511 1/20 0.59
CYP3A4 P08684 6/20 0.58
CYP1A2 P05177 3/20 0.58
CYP2C9 P11712 2/20 0.58
CYP2D6 P10635 1/20 0.58
CYP2C19 P33261 1/20 0.58
MAPT P10636 1/20 0.55
EGFR P00533 2/20 0.55
CYP2A6 P11509 1/20 0.54
NPC1 O15118 1/20 0.53
RAB9A P51151 1/20 0.53
PDGFRB P09619 2/20 0.51
PDGFRA P16234 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1204577 1.00 CYP11B2 (0.60) CYP11B2CYP11B1CYP17A1CYP19A1CYP3A4
SCHEMBL127857 0.94 CYP11B2 (0.58) CYP11B2CYP11B1CYP17A1CYP19A1CYP3A4
SCHEMBL7283560 0.85 CYP11B2 (0.61) CYP11B2CYP11B1CYP17A1CYP19A1CYP3A4
SCHEMBL15271125 0.83 RAB9A (0.51) CYP11B2CYP11B1CYP17A1CYP19A1CYP3A4
SCHEMBL25625872 0.83 CYP11B2 (0.53) CYP11B2CYP11B1CYP17A1CYP19A1CYP3A4
Ethyl Acetate SCHEMBL29093356 0.81 CYP3A4 (0.51) CYP11B2CYP11B1CYP3A4CYP1A2NPC1
SCHEMBL29447161 0.79 CYP1A2 (0.79) CYP11B2CYP11B1CYP3A4CYP1A2CYP2C9
SCHEMBL443070 0.79 CYP1A2 (0.79) CYP11B2CYP11B1CYP3A4CYP1A2CYP2C9
SCHEMBL1536335 0.79 PRKCZ (0.44) CYP11B2CYP11B1CYP17A1CYP19A1CYP3A4
SCHEMBL13302286 0.79 CYP11B1 (0.62) CYP11B2CYP11B1CYP19A1CYP1A2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4359388-A2 ISOQUINOLINE AND PYRIDINE BASED CXCR4 ANTAGONISTS Katholieke Universiteit Leuven (BE) 2024-05-01 EP disclosed
CN-116375740-A Difluoro pyrido [2,1-c ] [1,4] thiazine compounds and preparation method thereof 北京化工大学 2023-07-04 CN disclosed
WO-2022269027-A2 ISOQUINOLINE AND PYRIDINE BASED CXCR4 ANTAGONISTS KATHOLIEKE UNIVERSITEIT LEUVEN (BE) 2022-12-29 WO disclosed