SCHEMBL300665

SCHEMBL300665

C[C@H](NC(=O)Oc1n[nH]c2c1CCCC/C2=C\c1ccc(Cl)cc1)C1CCCCC1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 3/20 0.35
NPC1 O15118 1/20 0.35
HTT P42858 1/20 0.35
CNR1 P21554 6/20 0.35
CNR2 P34972 3/20 0.34
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34
HRH3 Q9Y5N1 2/20 0.34
P2RX7 Q99572 2/20 0.33
PRLHR P49683 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL300543 1.00 MAPK1 (0.35) MAPK1NPC1HTTCNR1CNR2
SCHEMBL176625 0.86 NPC1 (0.43) NPC1HTTCNR1CNR2TAS1R3
SCHEMBL176477 0.86 NPC1 (0.43) NPC1HTTCNR1CNR2TAS1R3
SCHEMBL300660 0.83 CNR1 (0.46) MAPK1CNR1CNR2
SCHEMBL300525 0.83 CNR1 (0.46) MAPK1CNR1CNR2
SCHEMBL300698 0.79 LIPE (0.48) NPC1HTTCNR1CNR2
SCHEMBL300451 0.78 CNR2 (0.42) MAPK1NPC1HTTCNR1CNR2
SCHEMBL300719 0.78 CNR1 (0.49) CNR1CNR2
SCHEMBL300714 0.78 CNR1 (0.48) CNR1CNR2
SCHEMBL300391 0.78 CNR1 (0.51) CNR1CNR2TAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937259-B1 HEXAHYDRO-CYCLOHEPTAPYRAZOLE CANNABINOID MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2011-11-23 EP claimed