SCHEMBL300698

SCHEMBL300698

O=C(NN1CCCCC1)Oc1n[nH]c2c1CCCC/C2=C\c1ccc(Cl)cc1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
LIPE Q05469 5/20 0.48
NPC1 O15118 1/20 0.38
HTT P42858 1/20 0.38
CNR1 P21554 8/20 0.37
PKM P14618 1/20 0.35
AKR1C3 P42330 1/20 0.34
AKR1C1 Q04828 1/20 0.34
CNR2 P34972 3/20 0.34
HDAC1 Q13547 1/20 0.34
PARP1 P09874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL300757 0.92 LIPE (0.49) LIPENPC1HTTCNR1
SCHEMBL176622 0.85 NPC1 (0.46) NPC1HTTCNR1CNR2
SCHEMBL176623 0.85 NPC1 (0.46) NPC1HTTCNR1CNR2
SCHEMBL300543 0.79 MAPK1 (0.35) NPC1HTTCNR1CNR2
SCHEMBL300665 0.79 MAPK1 (0.35) NPC1HTTCNR1CNR2
SCHEMBL300525 0.78 CNR1 (0.46) CNR1CNR2
SCHEMBL300660 0.78 CNR1 (0.46) CNR1CNR2
SCHEMBL176863 0.78 NPC1 (0.43) NPC1HTTAKR1C3AKR1C1
SCHEMBL176864 0.78 NPC1 (0.43) NPC1HTTAKR1C3AKR1C1
SCHEMBL176669 0.77 SMN1; SMN2 (0.46) LIPENPC1HTTCNR1AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937259-B1 HEXAHYDRO-CYCLOHEPTAPYRAZOLE CANNABINOID MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2011-11-23 EP claimed