SCHEMBL300693

SCHEMBL300693

O=C(NC1CCCC1)Oc1nn(C2CCCCC2)c2c1CCCCC2Cc1ccc(F)cc1

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 4/20 0.40
CNR2 P34972 4/20 0.40
EPHX1 P07099 1/20 0.39
CCR3 P51677 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL300549 0.86 THRB (0.41) CCR3POLB
SCHEMBL176414 0.84 NPC1 (0.44) CNR1CNR2CCR3POLB
SCHEMBL300546 0.84 VIPR2 (0.36) CNR1CNR2
SCHEMBL300472 0.84 PDE9A (0.38) CCR3POLB
SCHEMBL300365 0.83 CNR2 (0.41) CNR1CNR2
SCHEMBL176833 0.83 POLB (0.43) CNR1CNR2CCR3POLB
SCHEMBL300469 0.83 CYP3A4 (0.40) CNR2EPHX1
SCHEMBL300521 0.82 CNR2 (0.43) CNR2
SCHEMBL176941 0.82 NPC1 (0.41) CNR1CNR2CCR3POLB
SCHEMBL300474 0.79 EPHX2 (0.39) CNR2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937259-B1 HEXAHYDRO-CYCLOHEPTAPYRAZOLE CANNABINOID MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2011-11-23 EP claimed