SCHEMBL300472

SCHEMBL300472

O=C(NCc1ccc(C(F)(F)F)cc1)Oc1nn(C2CCCCC2)c2c1CCCCC2Cc1ccc(F)cc1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE9A O76083 2/20 0.38
POLB P06746 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TDP1 Q9NUW8 1/20 0.36
BTK Q06187 1/20 0.35
CCR3 P51677 2/20 0.35
P2RX7 Q99572 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL300549 0.91 THRB (0.41) POLBRAB9ASMN1; SMN2CCR3
SCHEMBL176656 0.86 ALDH1A1 (0.44) PDE9APOLBRAB9ASMN1; SMN2BTK
SCHEMBL300693 0.84 CNR1 (0.40) POLBCCR3
SCHEMBL300734 0.84 ALDH1A1 (0.38)
SCHEMBL300469 0.78 CYP3A4 (0.40)
SCHEMBL300521 0.77 CNR2 (0.43)
SCHEMBL300489 0.77 LPAR5 (0.41)
SCHEMBL300526 0.76 GLA (0.39) POLBRAB9ACCR3
SCHEMBL176706 0.76 THRB (0.47) POLBRAB9ASMN1; SMN2
SCHEMBL300546 0.76 VIPR2 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937259-B1 HEXAHYDRO-CYCLOHEPTAPYRAZOLE CANNABINOID MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2011-11-23 EP claimed