SCHEMBL300469

SCHEMBL300469

C[C@H](NC(=O)Oc1nn(C2CCCCC2)c2c1CCCCC2Cc1ccc(F)cc1)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
FKBP1A P62942 1/20 0.39
CACNA1G O43497 1/20 0.38
MAPK1 P28482 2/20 0.38
CNR2 P34972 1/20 0.37
EPHX1 P07099 2/20 0.36
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL300360 0.92 CNR2 (0.46) FKBP1AMAPK1CNR2EPHX1BCHE
SCHEMBL300521 0.90 CNR2 (0.43) CNR2
SCHEMBL300678 0.88 CNR2 (0.48) FKBP1AMAPK1CNR2
SCHEMBL176782 0.86 MAPK1 (0.45) CYP3A4CYP2D6CYP2C9CYP2C19FKBP1A
SCHEMBL300549 0.85 THRB (0.41) KDM4EALDH1A1
SCHEMBL300693 0.83 CNR1 (0.40) CNR2EPHX1
SCHEMBL176620 0.78 CNR2 (0.48) MAPK1CNR2ALDH1A1
SCHEMBL176638 0.78 CNR2 (0.48) MAPK1CNR2ALDH1A1
SCHEMBL300546 0.78 VIPR2 (0.36) CNR2
SCHEMBL300472 0.78 PDE9A (0.38)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937259-B1 HEXAHYDRO-CYCLOHEPTAPYRAZOLE CANNABINOID MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2011-11-23 EP claimed