SCHEMBL300757

SCHEMBL300757

O=C(NN1CCOCC1)Oc1n[nH]c2c1CCCC/C2=C\c1ccc(Cl)cc1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LIPE Q05469 9/20 0.49
SMN1; SMN2 Q16637 1/20 0.39
KDM4E B2RXH2 3/20 0.37
MAPT P10636 3/20 0.37
ALDH1A1 P00352 3/20 0.37
MAPK1 P28482 1/20 0.37
NPC1 O15118 2/20 0.36
HTT P42858 2/20 0.36
LMNA P02545 1/20 0.34
RAB9A P51151 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CNR1 P21554 1/20 0.34
TP53 P04637 1/20 0.34
MEN1 O00255 1/20 0.33
POLB P06746 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL300698 0.92 LIPE (0.48) LIPENPC1HTTCNR1
SCHEMBL176669 0.86 SMN1; SMN2 (0.46) LIPESMN1; SMN2KDM4EMAPTALDH1A1
SCHEMBL176670 0.86 SMN1; SMN2 (0.46) LIPESMN1; SMN2KDM4EMAPTALDH1A1
SCHEMBL300459 0.77 CNR2 (0.51) LIPEKDM4EMAPTCNR1MEN1
SCHEMBL176623 0.77 NPC1 (0.46) NPC1HTTCNR1
SCHEMBL176622 0.77 NPC1 (0.46) NPC1HTTCNR1
SCHEMBL300525 0.76 CNR1 (0.46) ALDH1A1MAPK1LMNAL3MBTL1CNR1
SCHEMBL300660 0.76 CNR1 (0.46) ALDH1A1MAPK1LMNAL3MBTL1CNR1
SCHEMBL300665 0.75 MAPK1 (0.35) MAPK1NPC1HTTCNR1
SCHEMBL300543 0.75 MAPK1 (0.35) MAPK1NPC1HTTCNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937259-B1 HEXAHYDRO-CYCLOHEPTAPYRAZOLE CANNABINOID MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2011-11-23 EP claimed