SCHEMBL30083006

SCHEMBL30083006

COc1ncc(Sc2c(Br)cc([N+](=O)[O-])cc2Br)cc1C(C)C

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.32
CRHBP P24387 1/20 0.32
HTT P42858 1/20 0.32
CRHR2 Q13324 1/20 0.32
PIK3CA P42336 1/20 0.32
HIF1A Q16665 1/20 0.32
EPAS1 Q99814 1/20 0.32
ALDH1A1 P00352 1/20 0.31
CYP3A4 P08684 1/20 0.31
LMNA P02545 1/20 0.31
IGF1R P08069 1/20 0.31
AMY1A P0DUB6 1/20 0.30
P2RX3 P56373 1/20 0.30
P2RX2 Q9UBL9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28660308 1.00 MAPT (0.32) MAPTCRHBPHTTCRHR2PIK3CA
SCHEMBL30083014 0.86 ALDH1A1 (0.35) MAPTHTTPIK3CAHIF1AEPAS1
SCHEMBL28664582 0.86 ALDH1A1 (0.35) MAPTHTTPIK3CAHIF1AEPAS1
SCHEMBL30083021 0.82 P2RX3 (0.38) MAPTPIK3CAP2RX3P2RX2
SCHEMBL30148695 0.77 ALDH1A1 (0.41) MAPTHTTALDH1A1LMNA
SCHEMBL30543269 0.71 MAPT (0.40) MAPTCRHBPHTTCRHR2ALDH1A1
SCHEMBL116509 0.71 MAPT (0.40) MAPTCRHBPHTTCRHR2ALDH1A1
SCHEMBL24449303 0.71 RORC (0.40) MAPTHTTALDH1A1LMNAAMY1A
SCHEMBL30083022 0.69 P2RX3 (0.35) MAPTPIK3CAP2RX3P2RX2
SCHEMBL24449302 0.69 RORC (0.41) MAPTHTTALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113698388-B 6-oxo-1, 6-dihydropyridine derivative, preparation method and application thereof in medicine 江苏恒瑞医药股份有限公司 2022-11-22 CN disclosed