SCHEMBL30083022

SCHEMBL30083022

COc1ncc(Sc2c(Cl)cc(N)cc2Cl)cc1C(C)C

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 5/20 0.35
P2RX2 Q9UBL9 5/20 0.35
AURKA O14965 1/20 0.34
TTK P33981 1/20 0.34
AURKB Q96GD4 1/20 0.34
INCENP Q9NQS7 1/20 0.34
PIK3R1 P27986 1/20 0.33
PIK3CA P42336 1/20 0.33
RORC P51449 2/20 0.32
MAPT P10636 1/20 0.32
CASP1 P29466 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30083021 0.84 P2RX3 (0.38) P2RX3P2RX2AURKATTKAURKB
SCHEMBL28664582 0.82 ALDH1A1 (0.35) PIK3CARORCMAPT
SCHEMBL30083014 0.82 ALDH1A1 (0.35) PIK3CARORCMAPT
SCHEMBL29527631 0.75 RORC (0.53) P2RX3P2RX2PIK3R1PIK3CARORC
SCHEMBL22959151 0.75 RORC (0.53) P2RX3P2RX2PIK3R1PIK3CARORC
SCHEMBL24449953 0.74 THRB (0.38) P2RX3P2RX2PIK3R1PIK3CARORC
SCHEMBL115578 0.73 PIK3R1 (0.40) P2RX3P2RX2AURKATTKAURKB
SCHEMBL24449964 0.70 RORC (0.46) P2RX3P2RX2PIK3R1PIK3CARORC
SCHEMBL11890406 0.70 TSHR (0.43) P2RX3P2RX2PIK3R1PIK3CARORC
SCHEMBL30083006 0.69 MAPT (0.32) P2RX3P2RX2PIK3CAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113698388-B 6-oxo-1, 6-dihydropyridine derivative, preparation method and application thereof in medicine 江苏恒瑞医药股份有限公司 2022-11-22 CN disclosed