SCHEMBL30101987

SCHEMBL30101987

CC(C)(O)Cc1nc2c(-c3cccnc3)nc(-c3ccc(C(F)(F)F)nc3)cc2c(=O)[nH]1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 3/20 0.37
PIM2 Q9P1W9 1/20 0.37
PTGS1 P23219 1/20 0.36
PTGS2 P35354 1/20 0.36
HSP90AA1 P07900 1/20 0.36
PTGES O14684 1/20 0.36
KCNH2 Q12809 1/20 0.35
SYK P43405 2/20 0.35
TRPV3 Q8NET8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30101920 0.90 PIM1 (0.38) PIM1PIM2PTGS1PTGS2KCNH2
SCHEMBL30101885 0.83 TRPV3 (0.40) PTGS1PTGS2PTGESKCNH2SYK
SCHEMBL30101836 0.83 TRPV3 (0.39) PTGS1PTGS2PTGESKCNH2SYK
SCHEMBL23390340 0.79 PIM1 (0.40) PIM1PTGS1PTGS2
SCHEMBL29611095 0.79 PIM1 (0.40) PIM1PTGS1PTGS2
SCHEMBL23390465 0.78 SYK (0.40) PIM1PTGS1PTGS2HSP90AA1KCNH2
SCHEMBL30101897 0.77 SYK (0.35) PIM1PTGS1PTGS2HSP90AA1KCNH2
SCHEMBL30101960 0.74 PIM1 (0.37) PIM1PIM2PTGS1PTGS2KCNH2
SCHEMBL30101994 0.74 PTGS2 (0.40) PIM1PIM2PTGS1PTGS2KCNH2
SCHEMBL23416810 0.74 CYP2E1 (0.41) PIM1PTGS1PTGS2HSP90AA1KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115443276-A Pyridopyrimidinone derivatives and their use as modulators of aromatic hydrocarbon receptors 东亚ST株式会社 2022-12-06 CN claimed
CN-115443276-A Pyridopyrimidinone derivatives and their use as modulators of aromatic hydrocarbon receptors 东亚ST株式会社 2022-12-06 CN disclosed