SCHEMBL30101994

SCHEMBL30101994

CS(=O)(=O)CCc1nc2c(-c3cccnc3)nc(-c3ccc(C(F)(F)F)cc3)cc2c(=O)[nH]1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.40
PTGS1 P23219 1/20 0.40
TRPV1 Q8NER1 1/20 0.38
PIM1 P11309 2/20 0.37
NPY5R Q15761 1/20 0.37
PIM2 Q9P1W9 1/20 0.37
DGAT1 O75907 1/20 0.37
KCNH2 Q12809 1/20 0.37
KIT P10721 2/20 0.35
TNKS O95271 3/20 0.35
TNKS2 Q9H2K2 3/20 0.35
PARP2 Q9UGN5 2/20 0.35
S1PR1 P21453 1/20 0.35
NPC1 O15118 1/20 0.34
PARP1 P09874 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
XBP1 P17861 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30101920 0.84 PIM1 (0.38) PTGS2PTGS1PIM1NPY5RPIM2
SCHEMBL31472806 0.83 XDH (0.41) PIM1MAPTL3MBTL1
SCHEMBL30101960 0.81 PIM1 (0.37) PTGS2PTGS1PIM1NPY5RPIM2
SCHEMBL31472805 0.80 PIM1 (0.39) PTGS2PTGS1PIM1NPY5RDGAT1
SCHEMBL30101909 0.79 AHR (0.39) PTGS2PTGS1PIM1NPY5RDGAT1
SCHEMBL30101887 0.79 PIM1 (0.39) PTGS2PTGS1PIM1NPY5RDGAT1
SCHEMBL23950293 0.78 PTGS2 (0.42) PTGS2PTGS1TRPV1PIM1NPY5R
SCHEMBL31472804 0.78 PIM1 (0.37) PTGS2PTGS1PIM1NPY5RDGAT1
SCHEMBL30101858 0.78 AHR (0.38) PTGS2PTGS1PIM1NPY5RDGAT1
SCHEMBL30101972 0.76 TNKS (0.50) PIM1NPY5RDGAT1KCNH2KIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115443276-A Pyridopyrimidinone derivatives and their use as modulators of aromatic hydrocarbon receptors 东亚ST株式会社 2022-12-06 CN claimed
CN-115443276-B Pyridopyrimidinone derivatives and their use as arene receptor modulators 东亚ST株式会社 2025-04-18 CN disclosed
CN-115443276-A Pyridopyrimidinone derivatives and their use as modulators of aromatic hydrocarbon receptors 东亚ST株式会社 2022-12-06 CN disclosed