SCHEMBL30102003

SCHEMBL30102003

CN1CCN(c2ccc(-c3cc4c(=O)[nH]c(CC(O)CO)nc4c(-c4cccnc4)n3)cc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TNKS O95271 2/20 0.39
PARP1 P09874 2/20 0.39
TNKS2 Q9H2K2 2/20 0.39
DYRK1A Q13627 3/20 0.39
CLK1 P49759 1/20 0.39
CHEK1 O14757 1/20 0.38
PIM1 P11309 2/20 0.38
MAP4K1 Q92918 2/20 0.37
CDK4 P11802 1/20 0.37
CCND1 P24385 1/20 0.37
CCND2 P30279 1/20 0.37
CCND3 P30281 1/20 0.37
ACVR1 Q04771 1/20 0.37
IRAK4 Q9NWZ3 1/20 0.37
SYK P43405 2/20 0.37
CLK2 P49760 1/20 0.37
CLK3 P49761 1/20 0.37
HTR6 P50406 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30101980 0.91 PIK3CB (0.40) DYRK1ACLK1PIM1IRAK4SYK
SCHEMBL30101960 0.82 PIM1 (0.37) TNKSPARP1TNKS2DYRK1APIM1
SCHEMBL23925581 0.80 SYK (0.42) DYRK1ACLK1PIM1CDK4CCND1
SCHEMBL30101871 0.78 PIK3CB (0.41) DYRK1ACLK1PIM1ACVR1IRAK4
SCHEMBL31472806 0.76 XDH (0.41) DYRK1ACLK1PIM1ACVR1SYK
SCHEMBL23925427 0.71 SYK (0.44) DYRK1ACLK1PIM1SYK
SCHEMBL30101911 0.69 JAK2 (0.40) DYRK1ACLK1PIM1SYKCLK2
SCHEMBL31472809 0.69 PIK3CA (0.48) DYRK1ACLK1PIM1SYK
SCHEMBL30101909 0.69 AHR (0.39) TNKSPARP1TNKS2PIM1
SCHEMBL30101920 0.69 PIM1 (0.38) TNKSPARP1TNKS2PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115443276-A Pyridopyrimidinone derivatives and their use as modulators of aromatic hydrocarbon receptors 东亚ST株式会社 2022-12-06 CN claimed
CN-115443276-A Pyridopyrimidinone derivatives and their use as modulators of aromatic hydrocarbon receptors 东亚ST株式会社 2022-12-06 CN disclosed