SCHEMBL30104016

SCHEMBL30104016

COC(=O)N1C[C@H](O[Si](C)(C)C(C)(C)C)C[C@H]1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.37
ATM Q13315 1/20 0.33
PPM1D O15297 1/20 0.32
UCHL1 P09936 1/20 0.31
KCNH2 Q12809 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3832181 0.88 UCHL1 (0.39) ATMPPM1DUCHL1
SCHEMBL29203075 0.88 UCHL1 (0.39) ATMPPM1DUCHL1
SCHEMBL18577100 0.88 UCHL1 (0.39) ATMPPM1DUCHL1
SCHEMBL239646 0.88 UCHL1 (0.39) ATMPPM1DUCHL1
SCHEMBL2809688 0.88 UCHL1 (0.39) ATMPPM1DUCHL1
SCHEMBL3832206 0.88 UCHL1 (0.39) ATMPPM1DUCHL1
SCHEMBL2708045 0.88 UCHL1 (0.39) ATMPPM1DUCHL1
SCHEMBL15203438 0.87 ATM (0.36) ATMPPM1D
SCHEMBL28776789 0.87 ATM (0.36) ATMPPM1D
SCHEMBL3528010 0.87 ATM (0.36) ATMPPM1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12630563-B2 Macrocyclic RIP2-kinase inhibitors ONCODESIGN S.A. (FR) 2026-05-19 US disclosed
US-20260125396-A1 MACROCYCLIC RIP2-KINASE INHIBITORS ONCODESIGN S.A. (FR) 2026-05-07 US disclosed
US-20240254140-A1 COMPOUNDS AND THEIR USE IN THE TREATMENT OF BACTERIAL INFECTION HOFFMANN-LA ROCHE INC. (US) 2024-08-01 US disclosed
US-20230126352-A1 MACROCYCLIC RIP2-KINASE INHIBITORS ONCODESIGN SA (FR) 2023-04-27 US disclosed
EP-4097110-A1 MACROCYCLIC RIP2-KINASE INHIBITORS Oncodesign S.A. (FR) 2022-12-07 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240254140-A1 COMPOUNDS AND THEIR USE IN THE TREATMENT OF BACTERIAL INFECTION C3AR1, LTB4R, C5 TSHR 1801/4885ATM 3666/4885PPM1D 3443/4885
US-20260125396-A1 MACROCYCLIC RIP2-KINASE INHIBITORS RIPK1, RIPK2, RIPK4 TSHR 1770/4885ATM 2809/4885PPM1D 903/4885
US-12630563-B2 Macrocyclic RIP2-kinase inhibitors RIPK1, RIPK2, RIPK3 TSHR 2985/4885ATM 2546/4885PPM1D 396/4885
US-20230126352-A1 MACROCYCLIC RIP2-KINASE INHIBITORS RIPK2, RIPK1, RIPK3 TSHR 3830/4885ATM 751/4885PPM1D 949/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.