SCHEMBL30107567

SCHEMBL30107567

COCCOc1cnc(Cl)nc1C#Cc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.41
PDGFRB P09619 1/20 0.39
PDGFRA P16234 1/20 0.39
EGFR P00533 1/20 0.38
GRM4 Q14833 1/20 0.36
VCP P55072 1/20 0.35
GRM5 P41594 4/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
TSHR P16473 1/20 0.35
POLB P06746 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
KCNH2 Q12809 1/20 0.34
EGLN1 Q9GZT9 1/20 0.33
ACACB O00763 1/20 0.33
PLAU P00749 1/20 0.33
ADK P55263 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28927186 1.00 FFAR1 (0.41) FFAR1PDGFRBPDGFRAEGFRGRM4
SCHEMBL28927139 0.84 GRM4 (0.41) PDGFRBPDGFRAEGFRGRM4TSHR
SCHEMBL30107565 0.75 ALDH1A1 (0.41) TSHRPLAU
SCHEMBL29197262 0.72 S1PR4 (0.41) TSHRPOLBL3MBTL1PLAU
SCHEMBL25430519 0.71 FFAR1 (0.46) FFAR1VCPGRM5L3MBTL1KCNH2
SCHEMBL30107573 0.71 MAPT (0.43) FFAR1GRM4GRM5PLAUADK
SCHEMBL17714326 0.71 ADK (0.44) FFAR1GRM4GRM5PLAUADK
SCHEMBL24047399 0.71 MAPT (0.43) FFAR1GRM4GRM5PLAUADK
SCHEMBL14976213 0.71 FFAR1 (0.42) FFAR1GRM4GRM5PLAUADK
SCHEMBL14232324 0.70 CHRNB2 (0.58) FFAR1ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4153577-A1 NEW MALONITRILE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2023-03-29 EP disclosed
CN-115551837-A Novel malononitrile derivatives 豪夫迈·罗氏有限公司 2022-12-30 CN disclosed