SCHEMBL13680584

SCHEMBL13680584

COC(=O)c1cccc(-c2cccc(C)n2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 1/20 0.53
GABRB3 P28472 1/20 0.53
GABRA5 P31644 1/20 0.53
GABRA3 P34903 1/20 0.53
CDK8 P49336 1/20 0.52
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA9 Q16790 1/20 0.50
SDHB P21912 1/20 0.50
ABL1 P00519 1/20 0.49
BCR P11274 1/20 0.49
SRC P12931 1/20 0.49
GRM5 P41594 2/20 0.49
PLAU P00749 2/20 0.49
ERN1 O75460 2/20 0.49
CYP2A6 P11509 1/20 0.49
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
LOXL2 Q9Y4K0 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680471 0.86 TDP1 (0.50) CA12CA1CA2CA9GRM5
SCHEMBL4895475 0.86 GABRG2 (0.66) GABRG2GABRB3GABRA5GABRA3CDK8
SCHEMBL6714723 0.83 CA12 (0.52) GABRG2GABRB3GABRA5GABRA3CDK8
SCHEMBL6718372 0.83 CNR1 (0.56) GABRG2GABRB3GABRA5GABRA3CDK8
SCHEMBL30107993 0.83 CDK8 (0.54) GABRG2GABRB3GABRA5GABRA3CDK8
SCHEMBL5557467 0.83 CDK8 (0.57) GABRG2GABRB3GABRA5GABRA3CDK8
SCHEMBL13680552 0.82 CYP2A6 (0.53) CDK8ABL1GRM5CYP2A6CCR1
SCHEMBL14189314 0.82 KMO (0.55) GRM5CYP2A6NPC1RAB9ACCR1
SCHEMBL8817643 0.82 PDE5A (0.53) GABRG2GABRB3GABRA5GABRA3GRM5
SCHEMBL16553302 0.81 GABRG2 (0.53) GABRG2GABRB3GABRA5GABRA3CDK8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed