SCHEMBL30108038

SCHEMBL30108038

COc1ccc2c(c1)nnn2-c1cc(N2CCC2)nc(N)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIM1 P11309 1/20 0.46
HRH4 Q9H3N8 4/20 0.45
KDM4E B2RXH2 4/20 0.42
ALDH1A1 P00352 4/20 0.42
SMN1; SMN2 Q16637 4/20 0.40
CRHBP P24387 1/20 0.40
CRHR2 Q13324 1/20 0.40
SCN2A Q99250 1/20 0.40
HPGD P15428 3/20 0.40
CYP1A2 P05177 2/20 0.40
CYP2C19 P33261 2/20 0.40
EZH2 Q15910 1/20 0.39
NUDT1 P36639 1/20 0.39
MEN1 O00255 3/20 0.38
KMT2A Q03164 3/20 0.38
HSD17B10 Q99714 2/20 0.38
USP2 O75604 1/20 0.38
LMNA P02545 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30108036 0.88 PIM1 (0.46) PIM1KDM4EALDH1A1SMN1; SMN2HPGD
SCHEMBL30107976 0.76 ROCK1 (0.34) HRH4KDM4EALDH1A1SMN1; SMN2SCN2A
SCHEMBL30107951 0.75 PTGS1 (0.46) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL30108003 0.73 MET (0.40) HRH4ALDH1A1HTTGAANPSR1
SCHEMBL30108039 0.73 ALDH1A1 (0.40) KDM4EALDH1A1SMN1; SMN2HPGDMEN1
SCHEMBL30107975 0.72 L3MBTL1 (0.40) PIM1KDM4EALDH1A1SMN1; SMN2MEN1
Hydrochloric Acid SCHEMBL29769980 0.70 FGFR1 (0.57) PIM1KDM4EALDH1A1SMN1; SMN2LMNA
Hydrochloric Acid SCHEMBL26907985 0.70 FGFR1 (0.57) PIM1KDM4EALDH1A1SMN1; SMN2LMNA
SCHEMBL31295948 0.68 SCN2A (0.74) HRH4KDM4ESCN2ACYP1A2CYP2C19
SCHEMBL30107966 0.68 TSHR (0.40) PIM1KDM4EALDH1A1SMN1; SMN2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022203399-A1 ADENOSINE A2A RECEPTOR ANTAGONIST AND USE THEREOF 주식회사 스탠다임 2022-09-29 WO disclosed