SCHEMBL30108042

SCHEMBL30108042

COCCOCc1cccc(Oc2ccc3c(c2)nnn3-c2cc(-c3ccco3)nc(N)n2)n1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 13/20 0.41
ADORA1 P30542 12/20 0.41
ADORA3 P0DMS8 8/20 0.41
ADORA2B P29275 8/20 0.41
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
UBE2I P63279 1/20 0.30
CACNA1B Q00975 1/20 0.30
APBA1 Q02410 1/20 0.30
SAE1 Q9UBE0 1/20 0.30
UBA2 Q9UBT2 1/20 0.30
MCL1 Q07820 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30107969 0.80 KDM4E (0.39) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL30107951 0.80 PTGS1 (0.46) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL30108028 0.78 KDM4E (0.43) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL30108055 0.78 ADORA2A (0.41) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL30108019 0.76 KEAP1 (0.39) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL30107980 0.75 ROCK1 (0.45) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL30107986 0.75 HSD17B10 (0.38) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL30107991 0.75 HSD17B10 (0.38) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL30107959 0.73 KDM4E (0.44) ADORA2AADORA1ADORA3ADORA2BKDM4E
SCHEMBL30108012 0.71 TSHR (0.58) ADORA2AADORA1ADORA3ADORA2BKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022203399-A1 ADENOSINE A2A RECEPTOR ANTAGONIST AND USE THEREOF 주식회사 스탠다임 2022-09-29 WO disclosed