SCHEMBL30108055

SCHEMBL30108055

COC(=O)c1cccc(-c2cccc(Oc3ccc4c(c3)nnn4-c3cc(-c4ccco4)nc(N)n3)n2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 9/20 0.41
ADORA1 P30542 9/20 0.41
ADORA3 P0DMS8 5/20 0.41
ADORA2B P29275 5/20 0.41
PTGS1 P23219 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.37
GRM5 P41594 1/20 0.34
POLB P06746 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
ESR1 P03372 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33
KMT2A Q03164 1/20 0.33
ESR2 Q92731 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ACSS2 Q9NR19 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30108019 0.92 KEAP1 (0.39) ADORA2AADORA1ADORA3ADORA2BPTGS1
SCHEMBL30107994 0.85 PTGS1 (0.50) ADORA2AADORA1ADORA3ADORA2BPTGS1
SCHEMBL30107969 0.81 KDM4E (0.39) ADORA2AADORA1ADORA3ADORA2BPTGS1
SCHEMBL30107951 0.79 PTGS1 (0.46) ADORA2AADORA1ADORA3ADORA2BPTGS1
SCHEMBL30108042 0.78 ADORA2A (0.41) ADORA2AADORA1ADORA3ADORA2BPTGS1
SCHEMBL30108028 0.77 KDM4E (0.43) ADORA2AADORA1ADORA3ADORA2BPTGS1
SCHEMBL30107998 0.76 ABL1 (0.34) ADORA2AADORA1KDM4EALDH1A1GAA
SCHEMBL30108023 0.74 PTGS1 (0.47) ADORA2AADORA1ADORA3ADORA2BPTGS1
SCHEMBL30107986 0.74 HSD17B10 (0.38) ADORA2AADORA1ADORA3ADORA2BPTGS1
SCHEMBL30107959 0.72 KDM4E (0.44) ADORA2AADORA1ADORA3ADORA2BKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022203399-A1 ADENOSINE A2A RECEPTOR ANTAGONIST AND USE THEREOF 주식회사 스탠다임 2022-09-29 WO disclosed