SCHEMBL30140434

SCHEMBL30140434

CC(C)(C)OC(=O)N1CC[C@H](Oc2nc3c(Nc4ccc(CC(F)(F)F)c(Cl)c4)ncnc3cc2F)C1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 1/20 0.47
PIK3CD O00329 10/20 0.45
EGFR P00533 6/20 0.43
ERBB2 P04626 3/20 0.43
EPHA2 P29317 2/20 0.43
EPHB4 P54760 2/20 0.43
PIK3CA P42336 2/20 0.43
PIK3CB P42338 2/20 0.43
PIK3CG P48736 2/20 0.43
KDR P35968 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30140320 0.89 EGFR (0.55) EGFRERBB2
SCHEMBL30140173 0.87 EGFR (0.47) GPR119PIK3CDEGFRERBB2EPHA2
SCHEMBL30140301 0.83 GPR119 (0.55) GPR119PIK3CDEGFRERBB2EPHB4
SCHEMBL23570650 0.83 GPR119 (0.52) GPR119PIK3CDEGFRERBB2EPHA2
SCHEMBL30140168 0.81 GPR119 (0.54) GPR119PIK3CDEGFRERBB2EPHB4
SCHEMBL30140077 0.80 PIK3CD (0.55) PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL30140184 0.80 GPR119 (0.55) GPR119PIK3CDEGFRPIK3CAPIK3CB
SCHEMBL30140092 0.79 GPR119 (0.57) GPR119PIK3CDEGFRERBB2PIK3CA
SCHEMBL30140252 0.79 GPR119 (0.52) GPR119PIK3CDEGFRERBB2PIK3CA
SCHEMBL30140382 0.79 EGFR (0.44) EGFRERBB2EPHA2EPHB4KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022266426-A1 6-(HETEROCYCLOALKYL-OXY)-QUINAZOLINE DERIVATIVES AND USES THEREOF BLACK DIAMOND THERAPEUTICS, INC. (US) 2022-12-22 WO disclosed